SCHEMBL14654152

SCHEMBL14654152

FC(F)(F)c1nc(-c2cccnc2)sc1-c1ccnc(-c2ncccn2)n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.45
ALOX5 P09917 1/20 0.45
RAB9A P51151 2/20 0.44
NPC1 O15118 1/20 0.44
CYP2A6 P11509 3/20 0.43
AXL P30530 1/20 0.40
PBRM1 Q86U86 1/20 0.40
MKNK1 Q9BUB5 1/20 0.40
MKNK2 Q9HBH9 1/20 0.40
HSP90AA1 P07900 1/20 0.40
HSP90AB1 P08238 1/20 0.40
PTK2 Q05397 1/20 0.40
HPGDS O60760 2/20 0.39
TRPM8 Q7Z2W7 1/20 0.38
MEN1 O00255 2/20 0.38
MAPT P10636 2/20 0.38
KMT2A Q03164 2/20 0.38
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 2/20 0.38
PTGS2 P35354 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14635624 0.91 ALOX5 (0.50) CYP19A1ALOX5RAB9ANPC1CYP2A6
SCHEMBL14654146 0.91 CYP2A6 (0.46) CYP19A1ALOX5RAB9ANPC1CYP2A6
SCHEMBL14654174 0.85 ALOX5 (0.41) CYP19A1ALOX5RAB9ANPC1CYP2A6
SCHEMBL15999643 0.85 CYP2A6 (0.53) CYP19A1ALOX5RAB9ANPC1CYP2A6
SCHEMBL1679855 0.82 CYP3A4 (0.49) CYP19A1ALOX5RAB9ANPC1CYP2A6
SCHEMBL14636146 0.79 ALOX5 (0.44) CYP19A1ALOX5RAB9ANPC1CYP2A6
SCHEMBL14636103 0.78 ALOX5 (0.41) CYP19A1ALOX5RAB9ANPC1CYP2A6
SCHEMBL15524984 0.76 PIK3CA (0.42) CYP19A1ALOX5RAB9ANPC1CYP2A6
SCHEMBL1679720 0.76 KDM4E (0.53) CYP19A1RAB9ANPC1CYP2A6AXL
SCHEMBL12279117 0.76 MEN1 (0.46) CYP19A1ALOX5RAB9ANPC1CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20140249024-A1 Pesticidal Methods Using Substituted 3-pyridyl Thiazole Compounds and Derivatives for Combating Animal Pests II BASF SE (DE) 2014-09-04 US disclosed
US-20140249024-A1 Pesticidal Methods Using Substituted 3-pyridyl Thiazole Compounds and Derivatives for Combating Animal Pests II BASF SE (DE) 2014-09-04 US disclosed
WO-2013010947-A2 PESTICIDAL METHODS USING SUBSTITUTED 3-PYRIDYL THIAZOLE COMPOUNDS AND DERIVATIVES FOR COMBATING ANIMAL PESTS II BASF SE (DE) 2013-01-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140249024-A1 Pesticidal Methods Using Substituted 3-pyridyl Thiazole Compounds and Derivatives for Combating Animal Pests II PTMS, PNPO, THOP1 CYP19A1 3049/4885ALOX5 1099/4885RAB9A 2297/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.