SCHEMBL146792

SCHEMBL146792

Cc1ccc(Cl)c(Cc2ccc(-c3ccc(N(C)C)cc3)s2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 5/20 0.42
SNCA P37840 2/20 0.38
TNF P01375 1/20 0.38
NOD1 Q9Y239 1/20 0.38
BCHE P06276 1/20 0.37
MEN1 O00255 1/20 0.37
NPC1 O15118 1/20 0.37
POLB P06746 1/20 0.37
RAB9A P51151 1/20 0.37
KMT2A Q03164 1/20 0.37
SLC5A2 P31639 5/20 0.37
SLC5A1 P13866 2/20 0.37
HSD17B1 P14061 6/20 0.36
HSD17B2 P37059 6/20 0.36
ALDH1A1 P00352 1/20 0.35
TSHR P16473 1/20 0.35
TDP1 Q9NUW8 1/20 0.34
SLC6A4 P31645 2/20 0.33
HTR2A P28223 1/20 0.33
KCNH2 Q12809 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9975462 0.84 HSD17B1 (0.46) APPSLC5A2SLC5A1HSD17B1HSD17B2
SCHEMBL14278458 0.84 CYP2A6 (0.45) MEN1NPC1RAB9AKMT2ASLC5A2
SCHEMBL147405 0.82 RORC (0.42) RAB9AKMT2ASLC5A2SLC5A1HSD17B1
SCHEMBL148158 0.81 CYP2A6 (0.37) MEN1NPC1POLBRAB9AKMT2A
SCHEMBL144713 0.80 SLC5A2 (0.41) RAB9AKMT2ASLC5A2SLC5A1HSD17B1
SCHEMBL148014 0.80 SLC5A2 (0.41) MEN1NPC1RAB9AKMT2ASLC5A2
SCHEMBL147396 0.79 APP (0.49) APPMEN1NPC1POLBRAB9A
SCHEMBL147481 0.79 SLC5A2 (0.40) SLC5A2SLC5A1HSD17B1HSD17B2SLC6A4
SCHEMBL156337 0.79 SLC5A2 (0.40) MEN1NPC1RAB9AKMT2ASLC5A2
SCHEMBL19677171 0.79 SLC5A2 (0.40) RAB9AKMT2ASLC5A2SLC5A1HSD17B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20160108078-A1 GLUCOPYRANOSIDE COMPOUND MITSUBISHI TANABE PHARMA CORPORATION (JP) 2016-04-21 US disclosed
US-20140296506-A1 GLUCOPYRANOSIDE COMPOUND MITSUBISHI TANABE PHARMA CORPORATION (JP) 2014-10-02 US disclosed
US-8785403-B2 Glucopyranoside compound MITSUBISHI TANABE PHARMA CORPORATION (JP) 2014-07-22 US disclosed
US-20120258913-A1 GLUCOPYRANOSIDE COMPOUND MITSUBISHI TANABE PHARMA CORPORATION (JP) 2012-10-11 US disclosed
US-8222219-B2 Glucopyranoside compound MITSUBISHI TANABE PHARMA CORPORATION (JP) 2012-07-17 US disclosed
US-8202984-B2 Glucopyranoside compound MITSUBISHI TANABE PHARMA CORPORATION (JP) 2012-06-19 US disclosed
US-20120058941-A1 GLUCOPYRANOSIDE COMPOUND MITSUBISHI TANABE PHARMA CORPORATION (JP) 2012-03-08 US disclosed
US-7943788-B2 Including the antidiabetic, antiobesity sodium glucose transport inhibitor Canagliflozin (1-( beta -D-glucopyranosyl)-4-methyl-3-[5-(4-fluorophenyl)-2-thienylmethyl]benzene) MITSUBISHI TANABE PHARMA CORPORATION (JP) 2011-05-17 US disclosed
US-20110105424-A1 GLUCOPYRANOSIDE COMPOUND MITSUBISHI TANABE PHARMA CORPORATION (JP) 2011-05-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120058941-A1 GLUCOPYRANOSIDE COMPOUND UGGT1, B3GAT3, FUT6 APP 2684/4885SNCA 3429/4885TNF 2224/4885
US-20110105424-A1 GLUCOPYRANOSIDE COMPOUND UGGT1, B3GAT3, FUT6 APP 2684/4885SNCA 3429/4885TNF 2224/4885
US-20120258913-A1 GLUCOPYRANOSIDE COMPOUND UGGT1, B3GAT3, FUT6 APP 2684/4885SNCA 3429/4885TNF 2224/4885
US-20160108078-A1 GLUCOPYRANOSIDE COMPOUND UGGT1, B3GAT3, FUT6 APP 2684/4885SNCA 3429/4885TNF 2224/4885
US-20140296506-A1 GLUCOPYRANOSIDE COMPOUND UGGT1, B3GAT3, FUT6 APP 2684/4885SNCA 3429/4885TNF 2224/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.