SCHEMBL14690185

SCHEMBL14690185

C[Si](C)(C)CCOCn1c(-c2ccccc2)nc(-c2ccncc2)c1-c1cccc(C(=O)O)c1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 3/20 0.41
CSNK1D P48730 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
TEK Q02763 3/20 0.39
TNK2 Q07912 1/20 0.39
NPC1 O15118 1/20 0.38
MAPT P10636 1/20 0.37
CSNK1E P49674 1/20 0.37
F11 P03951 1/20 0.37
PPARG P37231 1/20 0.36
FABP4 P15090 1/20 0.36
FABP5 Q01469 1/20 0.36
AKT1 P31749 2/20 0.36
AKT2 P31751 2/20 0.36
NR1H4 Q96RI1 1/20 0.36
EIF4EBP1 Q13541 1/20 0.36
ABCG2 Q9UNQ0 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14701090 0.92 MAPK14 (0.43) MAPK14MEN1KMT2ATEKF11
SCHEMBL16497631 0.91 MEN1 (0.45) MAPK14CSNK1DMEN1KMT2ATEK
SCHEMBL2148279 0.88 PIN1 (0.41) MAPK14MEN1KMT2ATEKMAPT
SCHEMBL2145931 0.85 TEK (0.39) MAPK14MEN1KMT2ATEKTNK2
SCHEMBL16497611 0.85 RAF1 (0.48) MAPK14MEN1KMT2ANPC1MAPT
SCHEMBL14701092 0.83 PDE4D (0.42) MEN1KMT2ATEKNPC1MAPT
SCHEMBL16497629 0.83 BRAF (0.44) MAPK14CSNK1DMEN1KMT2ATEK
SCHEMBL16510873 0.82 MEN1 (0.39) MAPK14MEN1KMT2ATEKTNK2
SCHEMBL16497623 0.82 MEN1 (0.40) MAPK14MEN1KMT2ATEKTNK2
SCHEMBL2148593 0.82 CYP1A2 (0.43) MAPK14MEN1KMT2ANPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130040983-A1 RAF KINASE INHIBITORS RUGA CORPORATION 2013-02-14 US disclosed
US-20130040983-A1 RAF KINASE INHIBITORS RUGA CORPORATION 2013-02-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130040983-A1 RAF KINASE INHIBITORS BRAF, RAF1, ARAF MAPK14 193/4885CSNK1D 531/4885MEN1 1820/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.