SCHEMBL14701090

SCHEMBL14701090

COC(=O)c1cccc(-c2c(-c3ccncc3)nc(-c3ccccc3)n2COCC[Si](C)(C)C)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 3/20 0.43
RAF1 P04049 1/20 0.42
ABCB1 P08183 1/20 0.42
ABCG2 Q9UNQ0 1/20 0.42
MGAM O43451 2/20 0.41
GAA P10253 2/20 0.41
SI P14410 2/20 0.41
MGAM2 Q2M2H8 2/20 0.41
DGAT1 O75907 1/20 0.40
TEK Q02763 3/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
F11 P03951 1/20 0.39
RIPK3 Q9Y572 1/20 0.38
NEK1 Q96PY6 1/20 0.38
ROCK2 O75116 1/20 0.37
PRKCA P17252 1/20 0.37
GRK2 P25098 1/20 0.37
TGFBR1 P36897 1/20 0.37
GSK3B P49841 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16497611 0.92 RAF1 (0.48) MAPK14RAF1MGAMGAASI
SCHEMBL14690185 0.92 MAPK14 (0.41) MAPK14ABCG2TEKMEN1KMT2A
SCHEMBL2148279 0.87 PIN1 (0.41) MAPK14MGAMGAASIMGAM2
SCHEMBL16497631 0.85 MEN1 (0.45) MAPK14RAF1TEKMEN1KMT2A
SCHEMBL2145931 0.83 TEK (0.39) MAPK14TEKMEN1KMT2AF11
SCHEMBL2148593 0.81 CYP1A2 (0.43) MAPK14GAAMEN1KMT2A
SCHEMBL14701092 0.81 PDE4D (0.42) GAATEKMEN1KMT2A
SCHEMBL16497629 0.81 BRAF (0.44) MAPK14TEKMEN1KMT2AF11
SCHEMBL16510873 0.80 MEN1 (0.39) MAPK14TEKMEN1KMT2AF11
SCHEMBL16497623 0.80 MEN1 (0.40) MAPK14TEKMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130040983-A1 RAF KINASE INHIBITORS RUGA CORPORATION 2013-02-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130040983-A1 RAF KINASE INHIBITORS BRAF, RAF1, ARAF MAPK14 193/4885RAF1 2/4885ABCB1 2086/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.