Alpha-Ketoglutaric Acid

Alpha-Ketoglutaric Acid

SCHEMBL1469844

NCCCCC(=O)O.O=C(O)CCC(=O)C(=O)O

nearest known ligand 0.73

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Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFKB1 P19838 2/20 0.73
CYP2D6 P10635 1/20 0.73
LMNA P02545 5/20 0.70
BLM P54132 2/20 0.70
NPSR1 Q6W5P4 2/20 0.70
THRB P10828 2/20 0.70
KMT2A Q03164 2/20 0.70
ALDH1A1 P00352 2/20 0.70
MEN1 O00255 1/20 0.70
PLG P00747 1/20 0.70
ALOX15 P16050 1/20 0.70
SLC6A2 P23975 1/20 0.70
RECQL P46063 1/20 0.70
SLC6A3 Q01959 1/20 0.70
EGLN1 Q9GZT9 2/20 0.64
MAPK1 P28482 1/20 0.64
SLC13A3 Q8WWT9 1/20 0.64
OR51E2 Q9H255 1/20 0.64
TSHR P16473 3/20 0.61
GABRR1 P24046 2/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Alpha-Ketoglutaric Acid SCHEMBL20817532 0.95 EGLN1 (0.70) NFKB1CYP2D6LMNABLMNPSR1
Alpha-Ketoglutaric Acid SCHEMBL16412456 0.93 LMNA (0.71) NFKB1CYP2D6LMNABLMNPSR1
Alpha-Ketoglutaric Acid SCHEMBL1469855 0.93 LMNA (0.71) NFKB1CYP2D6LMNABLMNPSR1
SCHEMBL728991 0.85 NFKB1 (0.62) NFKB1CYP2D6LMNABLMNPSR1
Adipic Acid SCHEMBL2537893 0.85 NFKB1 (1.00) NFKB1CYP2D6LMNABLMNPSR1
5-Aminovaleric Acid SCHEMBL190150 0.85
5-Aminovaleric Acid SCHEMBL887118 0.85 NFKB1 (1.00) NFKB1CYP2D6LMNABLMNPSR1
Alpha-Ketoglutaric Acid SCHEMBL1261453 0.83 EGLN1 (0.74) NFKB1CYP2D6LMNABLMNPSR1
SCHEMBL2368877 0.83 LMNA (0.64) NFKB1CYP2D6LMNABLMNPSR1
SCHEMBL285020 0.83 LMNA (0.64) NFKB1CYP2D6LMNABLMNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20190091300-A1 METHODS OF TREATING CANCER OF THE CENTRAL NERVOUS SYSTEM YEDA RESEARCH AND DEVELOPMENT CO. LTD. (IL) 2019-03-28 US disclosed
US-10159717-B2 Methods of treating cancer of the central nervous system YEDA RESEARCH AND DEVELOPMENT CO. LTD. (IL) 2018-12-25 US disclosed
US-20150216949-A1 METHODS OF TREATING CANCER OF THE CENTRAL NERVOUS SYSTEM YEDA RESEARCH AND DEVELOPMENT CO. LTD. (IL) 2015-08-06 US disclosed
US-9034319-B2 Methods of treating cancer of the central nervous system YEDA RESEARCH AND DEVELOPMENT CO. LTD. (IL) 2015-05-19 US disclosed
US-20110070218-A1 METHODS OF TREATING CANCER OF THE CENTRAL NERVOUS SYSTEM YEDA RESEARCH AND DEVELOPMENT CO. LTD. (IL) 2011-03-24 US disclosed
US-7767204-B2 Method and composition for protecting neuronal tissue from damage induced by elevated glutamate levels YEDA RESEARCH AND DEVELOPMENT CO. LTD. (IL) 2010-08-03 US disclosed
US-20090304661-A1 Method And Composition For Proctecting Neuronal Tissue From Damage Induced By Elevated Glutamate Levels YEDA RESEARCH AND DEVELOPMENT CO. LTD. AT THE WEIZMANN INSTITUTE OF SCEINCE (IL) 2009-12-10 US disclosed
US-20080233096-A1 transaminase, dehydrogenase, decarboxylase, ligase as glutamate modifying enzymes and oxaloacetate, pyruvate, NAD+, NADP+, 2-oxohexanedioic acid, 2-oxo-3-sulfopropionate, 2-oxo-3-sulfinopropionic acid, 2-oxo-3-phenylpropionic acid co-factors to enhance brain to blood efflux YEDA RESEARCH AND DEVELOPMENT CO. LTD. (IL) 2008-09-25 US disclosed
US-20080233099-A1 Method and composition for protecting neuronal tissue from damage induced by elevated glutamate levels YEDA RESEARCH AND DEVELOPMENT CO. LTD. (IL) 2008-09-25 US disclosed
US-7404951-B2 Method and composition for protecting neuronal tissue from damage induced by elevated glutamate levels YEDA RESEARCH AND DEVELOPMENT CO. LTD. (IL) 2008-07-29 US disclosed
US-20060024284-A1 Method and composition for protecting neuronal tissue from damage induced by elevated glutamate levels YEDA RESEARCH AND DEVELOPMENT CO. LTD. (IL) 2006-02-02 US disclosed