SCHEMBL14699641

SCHEMBL14699641

[N-]=[N+]=NCc1ccccc1C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FOLH1 Q04609 2/20 0.49
ALDH1A1 P00352 4/20 0.45
ALOX15 P16050 1/20 0.45
TSHR P16473 1/20 0.45
KAT2B Q92831 2/20 0.44
TP53 P04637 1/20 0.41
HTT P42858 1/20 0.41
HIF1A Q16665 2/20 0.40
GAA P10253 1/20 0.40
HMGB1 P09429 2/20 0.39
KDM4E B2RXH2 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
HPGD P15428 1/20 0.39
CA4 P22748 1/20 0.39
CA6 P23280 1/20 0.39
CA7 P43166 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CA9 Q16790 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26110049 0.87 FOLH1 (0.47) FOLH1ALDH1A1ALOX15TSHRKAT2B
SCHEMBL25408242 0.86 FOLH1 (0.58) FOLH1ALDH1A1ALOX15TSHRTP53
SCHEMBL28314204 0.85 KAT2B (0.38) FOLH1ALDH1A1ALOX15TSHRKAT2B
SCHEMBL15763694 0.84 KAT2B (0.40) ALDH1A1KAT2BKDM4EHPGDSMN1; SMN2
SCHEMBL14699642 0.84 KAT2B (0.40) FOLH1ALDH1A1ALOX15TSHRKAT2B
Hydrochloric Acid SCHEMBL29790654 0.83 KDM4E (0.40) ALDH1A1TSHRKAT2BGAAKDM4E
SCHEMBL28528967 0.81 FOLH1 (0.53) FOLH1ALDH1A1ALOX15TSHRHMGB1
SCHEMBL16588078 0.81 CTSD (0.46) ALDH1A1KAT2BGAACA1CA2
SCHEMBL10425173 0.81 FOLH1 (0.59) FOLH1ALDH1A1ALOX15TSHRTP53
SCHEMBL15353860 0.80 ALDH1A1 (0.53) ALDH1A1ALOX15TSHRHTTHIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 122 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4663205-A1 POLYMER-DRUG CONJUGATE, INTERMEDIATE THEREOF, AND USE THEREOF Shanghai Best-Link Bioscience, LLC (CN) 2025-12-17 EP claimed
US-20250340580-A1 TETRASACCHARIDES FOR THE DIAGNOSIS, PREVENTION, AND TREATMENT OF MELIOIDOSIS AND GLANDERS INST NAT RECH SCIENT (CA) 2025-11-06 US claimed
US-20250255977-A1 EPSILON-POLY-L-LYSINE-BASED DRUG CONJUGATE, INTERMEDIATE THEREOF, AND APPLICATION THEREOF SHANGHAI BEST-LINK BIOSCIENCE, LLC (CN) 2025-08-14 US claimed
WO-2025067481-A1 PHOSPHOLIPID DRUG CONJUGATE, AND PREPARATION METHOD AND USE THEREFOR 上海弼领生物技术有限公司 2025-04-03 WO claimed
WO-2024222960-A1 POLYMER-DRUG CONJUGATE, INTERMEDIATE THEREOF, AND USE THEREOF 上海弼领生物技术有限公司 2024-10-31 WO claimed
EP-4431116-A1 EPSILON-POLY-L-LYSINE-BASED DRUG CONJUGATE, INTERMEDIATE THEREOF, AND APPLICATION THEREOF Shanghai Best-Link Bioscience, LLC (CN) 2024-09-18 EP claimed
CN-118284435-A Drug conjugate based on epsilon-poly-L-lysine, intermediate and application thereof 上海弼领生物技术有限公司 2024-07-02 CN claimed
WO-2023078464-A1 EPSILON-POLY-L-LYSINE-BASED DRUG CONJUGATE, INTERMEDIATE THEREOF, AND APPLICATION THEREOF 上海弼领生物技术有限公司 2023-05-11 WO claimed
US-20230099200-A1 RADIOLABELED PEPTIDES FOR NON-INVASIVE DIAGNOSIS AND TREATMENT OF CXCR4 EXPRESSING TUMORS ISTITUTO NAZIONALE TUMORI IRCCS - FONDAZIONE G. PASCALE (IT) 2023-03-30 US claimed
EP-4081263-A1 RADIOLABELED PEPTIDES FOR NON-INVASIVE DIAGNOSIS AND TREATMENT OF CXCR4 EXPRESSING TUMORS Istituto Nazionale Tumori IRCCS - Fondazione G. Pascale (IT) 2022-11-02 EP claimed
US-20220227801-A1 TETRASACCHARIDES FOR THE DIAGNOSIS, PREVENTION, AND TREATMENT OF MELIOIDOSIS AND GLANDERS INSTITUT NATIONAL DE LA RECHERCHE EN SCIENTIFIQUE (CA) 2022-07-21 US claimed
EP-4007763-A1 TETRASACCHARIDES FOR THE DIAGNOSIS, PREVENTION, AND TREATMENT OF MELIOIDOSIS AND GLANDERS Institut National de la Recherche Scientifique (CA) 2022-06-08 EP claimed
WO-2021130329-A1 RADIOLABELED PEPTIDES FOR NON-INVASIVE DIAGNOSIS AND TREATMENT OF CXCR4 EXPRESSING TUMORS ISTITUTO NAZIONALE TUMORI IRCCS - FONDAZIONE G. PASCALE (IT) 2021-07-01 WO claimed
WO-2020243815-A1 TETRASACCHARIDES FOR THE DIAGNOSIS, PREVENTION, AND TREATMENT OF MELIOIDOSIS AND GLANDERS INSTITUT NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CA) 2020-12-10 WO claimed
CN-110003185-B Macrocyclic polyamine amphiphilic compound based on green fluorescent protein chromophore BI and preparation method and application thereof 北京师范大学 2020-05-19 CN claimed
EP-2727915-B1 Synthesis of deuterated catechols and benzo[d][1,3]dioxoles and derivatives thereof CONCERT PHARMACEUTICALS INC (US) 2016-04-13 EP claimed
EP-4234566-B1 MODIFIED NUCLEOSIDE OR NUCLEOTIDE BGI SHENZHEN (CN) 2026-04-15 EP disclosed
EP-4663205-A1 POLYMER-DRUG CONJUGATE, INTERMEDIATE THEREOF, AND USE THEREOF Shanghai Best-Link Bioscience, LLC (CN) 2025-12-17 EP disclosed
US-20090233280-A1 METHOD OF ACQUIRING INFORMATION REGARDING BASE SEQUENCE AND INFORMATION READING DEVICE FOR THE SAME CANON KABUSHIKI KAISHA (JP) 2009-09-17 US disclosed
WO-2007077952-A1 METHOD AND DEVICE FOR DETERMINING A NUCLEIC ACID ALLELE OR BASE SEQUENCE CANON KABUSHIKI KAISHA (JP) 2007-07-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250340580-A1 TETRASACCHARIDES FOR THE DIAGNOSIS, PREVENTION, AND TREATMENT OF MELIOIDOSIS AND GLANDERS NEU1, NEU4, NEU3 FOLH1 2966/4885ALDH1A1 3754/4885ALOX15 2393/4885
US-20230099200-A1 RADIOLABELED PEPTIDES FOR NON-INVASIVE DIAGNOSIS AND TREATMENT OF CXCR4 EXPRESSING TUMORS CXCR4, ACKR3, CXCL12 FOLH1 75/4885ALDH1A1 3650/4885ALOX15 4040/4885
US-20220227801-A1 TETRASACCHARIDES FOR THE DIAGNOSIS, PREVENTION, AND TREATMENT OF MELIOIDOSIS AND GLANDERS NEU1, NEU3, NEU4 FOLH1 2741/4885ALDH1A1 3702/4885ALOX15 2379/4885
US-20250255977-A1 EPSILON-POLY-L-LYSINE-BASED DRUG CONJUGATE, INTERMEDIATE THEREOF, AND APPLICATION THEREOF SLC7A1, KARS1, LNPEP FOLH1 347/4885ALDH1A1 1045/4885ALOX15 1431/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.