SCHEMBL1470282

SCHEMBL1470282

CCOC(=O)CCCc1ccc(N2Cc3ccc(F)cc3C2=O)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.41
CYP4Z1 Q86W10 2/20 0.40
CYP4F11 Q9HBI6 1/20 0.40
CYP4F12 Q9HCS2 1/20 0.40
BRD4 O60885 1/20 0.39
ALOX5 P09917 1/20 0.39
CYP4F2 P78329 1/20 0.38
CYP4A11 Q02928 1/20 0.38
TNF P01375 2/20 0.38
MAPK1 P28482 2/20 0.37
GAA P10253 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
RAB9A P51151 3/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
CASP3 P42574 1/20 0.37
HTR1A P08908 1/20 0.37
ADRA1A P35348 1/20 0.37
NPC1 O15118 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1467991 0.89 TNF (0.49) FAAHCYP4Z1CYP4F11CYP4F12BRD4
SCHEMBL1470284 0.86 CYP4Z1 (0.41) FAAHCYP4Z1CYP4F11CYP4F12BRD4
SCHEMBL1468613 0.85 CASP3 (0.45) FAAHCYP4Z1CYP4F11CYP4F12BRD4
SCHEMBL1467580 0.85 NPC1 (0.54) FAAHCYP4Z1CYP4F11CYP4F12ALOX5
SCHEMBL1467611 0.85 FFAR4 (0.45) MAPK1ADRA1A
SCHEMBL1468030 0.82 TNF (0.49) FAAHCYP4Z1CYP4F11CYP4F12BRD4
SCHEMBL1468193 0.80 CYP4Z1 (0.41) FAAHCYP4Z1CYP4F11CYP4F12BRD4
SCHEMBL1468434 0.79 CASP3 (0.45) FAAHCYP4Z1CYP4F11CYP4F12TNF
SCHEMBL5871481 0.76 CYP4F2 (0.58) FAAHCYP4Z1CYP4F11CYP4F12ALOX5
SCHEMBL1470394 0.73 GABRA1 (0.37) MAPK1GAARAB9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8722723-B2 Aromatic amide derivative RESEARCH FOUNDATION ITSUU LABORATORY (JP) 2014-05-13 US disclosed
US-20110071304-A1 AROMATIC AMIDE DERIVATIVE RESEARCH FOUNDATION ITSUU LABORATORY (JP) 2011-03-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110071304-A1 AROMATIC AMIDE DERIVATIVE NCOR2, NCOR1, EP300 FAAH 2385/4885CYP4Z1 963/4885CYP4F11 571/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.