SCHEMBL14709152

SCHEMBL14709152

O[C@H](CCl)c1ccc(Cl)s1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABBR2 O75899 1/20 0.43
GABBR1 Q9UBS5 1/20 0.43
GSK3B P49841 2/20 0.39
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
SLC6A3 Q01959 1/20 0.36
KCNH2 Q12809 1/20 0.36
TSHR P16473 1/20 0.35
TOP2A P11388 1/20 0.35
TOP2B Q02880 1/20 0.35
F2 P00734 1/20 0.34
DAO P14920 1/20 0.34
WRN Q14191 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
ALDH1A1 P00352 1/20 0.33
HTT P42858 1/20 0.33
RAB9A P51151 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27911200 1.00 GABBR2 (0.43) GABBR2GABBR1GSK3BCYP3A4CYP2D6
SCHEMBL21722781 0.83 GABBR2 (0.41) GABBR2GABBR1GSK3BCYP3A4CYP2D6
SCHEMBL21722780 0.83 GABBR2 (0.41) GABBR2GABBR1GSK3BCYP3A4CYP2D6
SCHEMBL5250926 0.83 GABBR2 (0.43) GABBR2GABBR1GSK3BCYP3A4CYP2D6
SCHEMBL5247316 0.83 GABBR2 (0.43) GABBR2GABBR1GSK3BCYP3A4CYP2D6
SCHEMBL5246292 0.83 GABBR2 (0.43) GABBR2GABBR1GSK3BCYP3A4CYP2D6
SCHEMBL22585593 0.81 GABBR2 (0.42) GABBR2GABBR1GSK3BCYP3A4CYP2D6
SCHEMBL17459297 0.81 GABBR2 (0.54) GABBR2GABBR1GSK3BCYP3A4CYP2D6
SCHEMBL9522198 0.77 TOP2A (0.45) GABBR2GABBR1GSK3BCYP3A4CYP2D6
SCHEMBL31378989 0.76 GABBR2 (0.42) GABBR2GABBR1GSK3BCYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013023511-A1 TRIAZOLOPYRIMIDINE DERIVATIVE AND PREPARATION METHOD AND USE THEREOF 上海恒瑞医药有限公司 (CN) 2013-02-21 WO disclosed
CN-102924457-A Triazolopyrimidine derivatives, preparation method and uses thereof SHANGHAI HENGRUI PHARM CO LTD 2013-02-13 CN disclosed