SCHEMBL14714005

SCHEMBL14714005

O=[N+]([O-])c1cc(CBr)[nH]n1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.30
MAPT P10636 2/20 0.30
KMT2A Q03164 2/20 0.30
NPC1 O15118 1/20 0.30
POLB P06746 1/20 0.30
PKM P14618 1/20 0.30
RAB9A P51151 1/20 0.30
MCL1 Q07820 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
APOBEC3G Q9HC16 1/20 0.30
ALDH1A1 P00352 2/20 0.30
KDM4E B2RXH2 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
ALOX15 P16050 1/20 0.30
TSHR P16473 1/20 0.30
MAPK1 P28482 1/20 0.30
NOS1 P29475 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12200985 0.81 HCAR2 (0.46) MEN1MAPTKMT2APOLBMCL1
SCHEMBL173914 0.81 HCAR2 (0.47) MAPTPOLBPKMALDH1A1KDM4E
SCHEMBL31319635 0.78 HCAR2 (0.49) APOBEC3GALDH1A1KDM4ETSHRCYP2C19
SCHEMBL16622728 0.78 LMNA (0.35)
SCHEMBL27683382 0.77 CYP1A2 (0.38) MEN1MAPTKMT2AALDH1A1KDM4E
SCHEMBL28079252 0.74 HCAR2 (0.32)
SCHEMBL3582886 0.74
SCHEMBL2427435 0.74
SCHEMBL10399847 0.73 HCAR2 (0.54) ALDH1A1
SCHEMBL28262261 0.71

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013024078-A1 INHIBITORS OF BRUTON'S TYROSINE KINASE F. HOFFMANN-LA ROCHE AG (CH) 2013-02-21 WO disclosed