SCHEMBL14715685

SCHEMBL14715685

NC(=O)[C@H]1CC[C@H](CCN2CCC(Oc3c(F)cc(F)cc3F)CC2)CC1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 1/20 0.38
SMN1; SMN2 Q16637 3/20 0.37
HRH1 P35367 1/20 0.37
CCR3 P51677 1/20 0.37
ALDH1A1 P00352 2/20 0.37
NAMPT P43490 1/20 0.37
NPSR1 Q6W5P4 1/20 0.36
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36
MAPK1 P28482 1/20 0.36
HIF1A Q16665 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
CACNA1I Q9P0X4 1/20 0.36
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3959814 1.00 OPRK1 (0.38) OPRK1SMN1; SMN2HRH1CCR3ALDH1A1
SCHEMBL3959816 0.89 CACNA1I (0.42) HRH1CCR3ALDH1A1CACNA1IPOLB
SCHEMBL14715704 0.89 CACNA1I (0.42) HRH1CCR3ALDH1A1CACNA1IPOLB
SCHEMBL14715697 0.87 HRH1 (0.46) SMN1; SMN2HRH1CCR3ALDH1A1
SCHEMBL3963825 0.87 HRH1 (0.46) SMN1; SMN2HRH1CCR3ALDH1A1
SCHEMBL3093392 0.84 DRD2 (0.39) NAMPTCACNA1I
SCHEMBL3959818 0.84 DRD2 (0.39) NAMPTCACNA1I
SCHEMBL3959812 0.84 HRH1 (0.39) OPRK1SMN1; SMN2HRH1CCR3NAMPT
SCHEMBL14715671 0.84 HRH1 (0.39) OPRK1SMN1; SMN2HRH1CCR3NAMPT
SCHEMBL3969152 0.83 NAMPT (0.48) OPRK1HRH1CCR3NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079693-B1 ETHER DERIVATIVES DUAL MODULATORS OF THE 5-HT2A AND D3 RECEPTORS HOFFMANN LA ROCHE (CH) 2013-02-27 EP claimed