SCHEMBL3093392

SCHEMBL3093392

N[C@H]1CC[C@H](CCN2CCC(Oc3c(F)cc(F)cc3F)CC2)CC1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 3/20 0.39
HTR1A P08908 1/20 0.37
HTR2A P28223 1/20 0.37
DRD3 P35462 1/20 0.37
NAMPT P43490 1/20 0.33
GRM2 Q14416 1/20 0.33
SLC6A4 P31645 1/20 0.33
FPR2 P25090 1/20 0.32
PROKR1 Q8TCW9 1/20 0.32
CACNA1I Q9P0X4 1/20 0.32
GPR6 P46095 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3959818 1.00 DRD2 (0.39) DRD2HTR1AHTR2ADRD3NAMPT
SCHEMBL3086254 0.88 DRD2 (0.46) DRD2HTR1AHTR2ADRD3CACNA1I
SCHEMBL3967377 0.88 DRD2 (0.46) DRD2HTR1AHTR2ADRD3CACNA1I
SCHEMBL14715685 0.84 OPRK1 (0.38) NAMPTCACNA1I
SCHEMBL3959814 0.84 OPRK1 (0.38) NAMPTCACNA1I
SCHEMBL3086252 0.84 GRM2 (0.47) DRD2GRM2SLC6A4GPR6
SCHEMBL14715699 0.84 GRM2 (0.47) DRD2GRM2SLC6A4GPR6
SCHEMBL3963647 0.82 DRD2 (0.39) DRD2HTR1AHTR2ADRD3NAMPT
SCHEMBL3087227 0.82 DRD2 (0.39) DRD2HTR1AHTR2ADRD3NAMPT
SCHEMBL3067860 0.81 HTR7 (0.46) DRD2HTR2ANAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079693-B1 ETHER DERIVATIVES DUAL MODULATORS OF THE 5-HT2A AND D3 RECEPTORS HOFFMANN LA ROCHE (CH) 2013-02-27 EP claimed
US-7795437-B2 Ether derivatives HOFFMANN-LA ROCHE INC. (US) 2010-09-14 US disclosed