Perazine

Perazine

SCHEMBL147165

CN1CCN(CCCN2c3ccccc3Sc3ccccc32)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 13/20 1.00
HTR1A P08908 4/20 0.78
ADRA2A P08913 4/20 0.78
CHRM1 P11229 4/20 0.78
DRD2 P14416 4/20 0.78
ADRA2C P18825 4/20 0.78
DRD1 P21728 4/20 0.78
SLC6A2 P23975 4/20 0.78
HTR2A P28223 4/20 0.78
SLC6A4 P31645 4/20 0.78
ADRA1A P35348 4/20 0.78
HRH1 P35367 4/20 0.78
DRD3 P35462 4/20 0.78
SLC6A3 Q01959 4/20 0.78
KCNH2 Q12809 4/20 0.78
LMNA P02545 3/20 0.78
TP53 P04637 3/20 0.78
CYP3A4 P08684 3/20 0.78
ADORA3 P0DMS8 3/20 0.78
MAPT P10636 3/20 0.78

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Perazine SCHEMBL29390464 1.00 KDM1A (1.00) KDM1AHTR1AADRA2ACHRM1DRD2
Perazine SCHEMBL6644457 0.98 KDM1A (0.97) KDM1AHTR1AADRA2ACHRM1DRD2
Perazine SCHEMBL2237726 0.98 KDM1A (0.97) KDM1AHTR1AADRA2ACHRM1DRD2
SCHEMBL6859184 0.97 KDM1A (0.94) KDM1AHTR1AADRA2ACHRM1DRD2
Perazine SCHEMBL10531680 0.92 KDM1A (0.84) KDM1AHTR1AADRA2ACHRM1DRD2
SCHEMBL10973127 0.91 KDM1A (0.84) KDM1AHTR1AADRA2ACHRM1DRD2
SCHEMBL2615404 0.89 KDM1A (0.80) KDM1AHTR1AADRA2ACHRM1DRD2
Perazine SCHEMBL7654455 0.88 CYP3A4 (0.82) KDM1AHTR1AADRA2ACHRM1DRD2
SCHEMBL7594811 0.88 KDM1A (0.78) KDM1AHTR1AADRA2ACHRM1DRD2
SCHEMBL2548635 0.88 KDM1A (0.78) KDM1AHTR1AADRA2ACHRM1DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2873 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3607938-B1 PHARMACEUTICAL COMPOSITION SOVIC BRKICIC LJILJANA (HR) 2026-05-27 EP claimed
EP-3507371-B1 COMPOSITIONS FOR TREATING DISEASES AND DISORDERS OF THE NERVOUS SYSTEM UNIV RUTGERS (US) 2026-01-28 EP claimed
US-12527754-B2 Methods and compositions for preventing and treating metabolic syndrome induced by antipsychotic treatment and related diseases and conditions TUFTS MEDICAL CENTER, INC. (US) 2026-01-20 US claimed
EP-4618973-A1 METHODS OF SWITCHING NEUROPSYCHIATRIC MEDICATIONS USING ULOTARONT Sumitomo Pharma America, Inc. (US) 2025-09-24 EP claimed
US-20250179064-A1 BENZOQUINOLONE INHIBITORS OF VMAT2 AUSPEX PHARMACEUTICALS LLC 2025-06-05 US claimed
WO-2025101418-A1 TREATMENT OF PSYCHIATRIC OR NEUROLOGICAL DISORDERS IN PATIENTS WITH PROMINENT ANHEDONIA USING IRDABISANT AS A MONOTHERAPY OR IN COMBINATION WITH AN ANTIPSYCHOTIC AGENT ALTO NEUROSCIENCE, INC. (US) 2025-05-15 WO claimed
US-20250144092-A1 TREATMENT OF PSYCHIATRIC OR NEUROLOGICAL DISORDERS IN PATIENTS WITH PROMINENT ANHEDONIA USING IRDABISANT AS A MONOTHERAPY OR IN COMBINATION WITH AN ANTIPSYCHOTIC AGENT ALTO NEUROSCIENCE, INC. 2025-05-08 US claimed
WO-2024107681-A1 METHODS OF SWITCHING NEUROPSYCHIATRIC MEDICATIONS USING ULOTARONT SUMITOMO PHARMA AMERICA, INC. (US) 2024-05-23 WO claimed
US-20240000810-A1 USE OF CANNABINOIDS IN THE TREATMENT OF TOURETTE SYNDROME AND TIC DISORDERS Orcosa Inc. (US) 2024-01-04 US claimed
EP-3192499-B1 CELLULOSE FIBRE BASED SUPPORT MATRICES FOR LAYERED PRODUCTS FOR ORAL AND PERORAL APPLICATION AND THEIR PREPARATION GLATT GMBH (DE) 2023-11-29 EP claimed
US-5785976-A Solid lipid particles, particles of bioactive agents and methods for the manufacture and use thereof PHARMACIA & UPJOHN AB (SE) 1998-07-28 US claimed
EP-0738257-A1 NEW METHOD FOR N-CYCLOPROPYLATION OF AROMATIC AMINES, AS WELL AS COMPOUNDS AND COMPOSITIONS OBTAINED SOMFAI, Eva, Dr. (HU) 1996-10-23 EP claimed
EP-0707637-A1 ENHANCEMENT OF LACCASE REACTIONS NOVO NORDISK A/S (DK) 1996-04-24 EP claimed
EP-0687172-A1 SOLID LIPID PARTICLES, PARTICLES OF BIOACTIVE AGENTS AND METHODS FOR THE MANUFACTURE AND USE THEREOF Pharmacia & Upjohn Aktiebolag (SE) 1995-12-20 EP claimed
EP-0679183-A1 ENHANCEMENT OF ENZYME REACTIONS NOVO NORDISK A/S (DK) 1995-11-02 EP claimed
CN-1110605-A Method of treating fungal infections LILLY CO ELI (US) 1995-10-25 CN claimed
WO-1995002573-A2 NEW METHOD FOR N-CYCLOPROPYLATION OF AROMATIC AMINES, AS WELL AS COMPOUNDS AND COMPOSITIONS OBTAINED SOMFAI EVA (HU) 1995-01-26 WO claimed
WO-1995001426-A1 ENHANCEMENT OF LACCASE REACTIONS NOVO NORDISK A/S (DK) 1995-01-12 WO claimed
WO-1994020072-A1 SOLID LIPID PARTICLES, PARTICLES OF BIOACTIVE AGENTS AND METHODS FOR THE MANUFACTURE AND USE THEREOF PHARMACIA AB (SE) 1994-09-15 WO claimed
WO-1994012621-A1 ENHANCEMENT OF ENZYME REACTIONS NOVO NORDISK (DK) 1994-06-09 WO claimed