SCHEMBL14718585

SCHEMBL14718585

CC(C)(C)OC(=O)N1CC(=O)C(c2ccccc2)=C(c2ccccc2)C1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
USP30 Q70CQ3 6/20 0.47
GPR119 Q8TDV5 1/20 0.43
CKS1B P61024 2/20 0.43
SKP1 P63208 2/20 0.43
SKP2 Q13309 2/20 0.43
MAPK1 P28482 1/20 0.42
SCD5 Q86SK9 1/20 0.41
PTGS1 P23219 1/20 0.40
PTGS2 P35354 1/20 0.40
NR1H2 P55055 1/20 0.40
EGFR P00533 1/20 0.39
SRC P12931 1/20 0.39
KDM4E B2RXH2 1/20 0.39
PKM P14618 1/20 0.39
NAMPT P43490 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14719295 0.86 USP30 (0.44) USP30GPR119CKS1BSKP1SKP2
SCHEMBL14719212 0.83 SCD5 (0.43) USP30GPR119CKS1BSKP1SKP2
SCHEMBL1751366 0.81 GPR119 (0.45) USP30GPR119CKS1BSKP1SKP2
SCHEMBL14719326 0.77 USP30 (0.40) USP30GPR119CKS1BSKP1SKP2
SCHEMBL31080015 0.75 USP2 (0.50) GPR119MAPK1NR1H2KDM4E
SCHEMBL1751873 0.75 ESR2 (0.48) USP30GPR119CKS1BSKP1SKP2
SCHEMBL1751837 0.74 CHRM5 (0.53) CKS1BSKP1SKP2
SCHEMBL17369314 0.73 MAPK1 (0.54) GPR119MAPK1NR1H2NAMPT
SCHEMBL29813840 0.73 MAPK1 (0.54) GPR119MAPK1NR1H2NAMPT
SCHEMBL16049290 0.73 ESR2 (0.46) USP30GPR119CKS1BSKP1SKP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130053565-A1 SUBSTITUTED 3-PIPERIDONE COMPOUNDS UNIVERSITY OF UTAH RESEARCH FOUNDATION (US) 2013-02-28 US disclosed
US-20130053565-A1 SUBSTITUTED 3-PIPERIDONE COMPOUNDS UNIVERSITY OF UTAH RESEARCH FOUNDATION (US) 2013-02-28 US disclosed
US-20130053565-A1 SUBSTITUTED 3-PIPERIDONE COMPOUNDS UNIVERSITY OF UTAH RESEARCH FOUNDATION (US) 2013-02-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130053565-A1 SUBSTITUTED 3-PIPERIDONE COMPOUNDS HTR3C, NPEPPS, RAP2C USP30 3130/4885GPR119 1675/4885CKS1B 2001/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.