SCHEMBL14720178

SCHEMBL14720178

NC(=O)Cc1c(F)cc(Br)cc1F

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 1/20 0.46
GPR17 Q13304 1/20 0.39
HTT P42858 1/20 0.34
PLA2G2A P14555 1/20 0.34
CA2 P00918 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
TAAR1 Q96RJ0 1/20 0.33
SIRT1 Q96EB6 1/20 0.33
LMNA P02545 1/20 0.33
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2566904 0.83 CES2 (0.40) GPR17HTTCA2TAAR1
SCHEMBL4928410 0.81 GPR17 (0.43) DGAT1GPR17LMNAMEN1KMT2A
SCHEMBL30749073 0.79 MAPT (0.35) DGAT1GPR17SMN1; SMN2SIRT1LMNA
SCHEMBL4925355 0.79 DGAT1 (0.37) DGAT1GPR17HTTSMN1; SMN2LMNA
SCHEMBL3261013 0.76 SIRT1 (0.39) DGAT1GPR17HTTSIRT1MEN1
SCHEMBL1317647 0.76 DGAT1 (0.55) DGAT1GPR17CA2SMN1; SMN2LMNA
SCHEMBL31551664 0.75 DGAT1 (0.55) DGAT1SIRT1MEN1KMT2A
SCHEMBL538344 0.75 DGAT1 (0.55) DGAT1SIRT1MEN1KMT2A
SCHEMBL22830383 0.75 HSP90AB1 (0.43) DGAT1SMN1; SMN2LMNAMEN1KMT2A
SCHEMBL31310136 0.75 GPR17 (0.39) DGAT1GPR17CA2LMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4565588-A1 BIOLOGICALLY ACTIVE COMPOUNDS AND METHODS THEREOF Suzhou Keen Therapeutics Co., Ltd. (CN) 2025-06-11 EP disclosed
WO-2023241620-A1 BIOLOGICALLY ACTIVE COMPOUNDS AND METHODS THEREOF SUZHOU KEEN THERAPEUTICS CO., LTD. (CN) 2023-12-21 WO disclosed
CN-113382991-B Aminopyrimidines useful for inhibiting protein tyrosine kinase activity 深圳市塔吉瑞生物医药有限公司 2022-12-27 CN disclosed
EP-2744333-B1 FATTY ACID SYNTHASE INHIBITORS GLAXOSMITHKLINE IP NO 2 LTD (GB) 2016-10-05 EP disclosed
US-9084794-B2 Fatty acid synthase inhibitors GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO. 2) LIMITED (GB) 2015-07-21 US disclosed
US-20140194415-A1 FATTY ACID SYNTHASE INHIBITORS GlaxoSmithKline Intellectual Property (No2) Limite (GB) 2014-07-10 US disclosed
EP-2744333-A1 FATTY ACID SYNTHASE INHIBITORS Glaxosmithkline Intellectual Property (No. 2) Limited (GB) 2014-06-25 EP disclosed
WO-2013028447-A1 FATTY ACID SYNTHASE INHIBITORS GLAXOSMITHKLINE LLC (US) 2013-02-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140194415-A1 FATTY ACID SYNTHASE INHIBITORS FASN, FADS2, FADS1 DGAT1 93/4885GPR17 515/4885HTT 4551/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.