SCHEMBL14720311

SCHEMBL14720311

OC1CC(N2CCC(=Cc3ccc(Br)cc3)CC2)C1

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 8/20 0.38
SRD5A2 P31213 4/20 0.35
ALDH1A1 P00352 1/20 0.33
L3MBTL3 Q96JM7 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
GPR183 P32249 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
HRH3 Q9Y5N1 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14721035 0.85 MCHR1 (0.36) MCHR1SRD5A2L3MBTL3L3MBTL1RAB9A
SCHEMBL14720608 0.81 HRH3 (0.43) MCHR1SRD5A2L3MBTL3L3MBTL1GPR183
SCHEMBL14720920 0.81 HRH3 (0.47) MCHR1SRD5A2L3MBTL3L3MBTL1GPR183
SCHEMBL14722284 0.78 HRH3 (0.44) MCHR1SRD5A2L3MBTL3L3MBTL1GPR183
SCHEMBL14722836 0.78 HRH3 (0.41) MCHR1SRD5A2L3MBTL3L3MBTL1GPR183
SCHEMBL14720913 0.75 GPR183 (0.38) MCHR1SRD5A2ALDH1A1L3MBTL3L3MBTL1
SCHEMBL14722992 0.74 MCHR1 (0.33) MCHR1
SCHEMBL12891140 0.72 MAOA (0.45) ALDH1A1RAB9A
SCHEMBL14720631 0.71 HRH3 (0.45) MCHR1SRD5A2GPR183NPC1RAB9A
SCHEMBL22804454 0.70 SLC18A3 (0.44) ALDH1A1HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013027001-A1 COMPOUNDS AND THEIR USE TO TREAT HISTAMINE H3 RELATED DISORDERS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-02-28 WO disclosed
WO-2013027001-A1 COMPOUNDS AND THEIR USE TO TREAT HISTAMINE H3 RELATED DISORDERS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-02-28 WO disclosed