SCHEMBL14720490

SCHEMBL14720490

C(=C1CCN(C2CCC2)CC1)c1ccc(COc2cccnc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 9/20 0.49
CYP2D6 P10635 2/20 0.46
MAPT P10636 1/20 0.42
RAB9A P51151 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
CHRNB2 P17787 2/20 0.41
CHRNA4 P43681 2/20 0.41
CHRNA1 P02708 1/20 0.41
CHRNB1 P11230 1/20 0.41
CHRNB4 P30926 1/20 0.41
CHRNA3 P32297 1/20 0.41
CHRNA7 P36544 1/20 0.41
CHRNB3 Q05901 1/20 0.41
CSF1R P07333 1/20 0.39
TRPV6 Q9H1D0 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14720972 0.82 HRH3 (0.42) HRH3CYP2D6
SCHEMBL14720482 0.79 RAB9A (0.46) HRH3CYP2D6RAB9ACSF1RTRPV6
SCHEMBL14721216 0.75 HRH3 (0.40) HRH3CYP2D6
SCHEMBL14720398 0.73 HRH3 (0.45) HRH3CYP2D6CHRNB2CHRNA4CHRNB1
SCHEMBL14720755 0.73 HRH3 (0.40) HRH3CYP2D6RAB9A
SCHEMBL14720672 0.73 HRH3 (0.38) HRH3CYP2D6
SCHEMBL14721067 0.72 SRD5A2 (0.42) HRH3CYP2D6
SCHEMBL3098064 0.72 HRH3 (0.75) HRH3CYP2D6
SCHEMBL14721508 0.71 HRH3 (0.38) HRH3CYP2D6
SCHEMBL14720592 0.71 HRH3 (0.35) HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013027001-A1 COMPOUNDS AND THEIR USE TO TREAT HISTAMINE H3 RELATED DISORDERS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-02-28 WO claimed
WO-2013027001-A1 COMPOUNDS AND THEIR USE TO TREAT HISTAMINE H3 RELATED DISORDERS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-02-28 WO disclosed
WO-2013027001-A1 COMPOUNDS AND THEIR USE TO TREAT HISTAMINE H3 RELATED DISORDERS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-02-28 WO disclosed