Quinoline

Quinoline

SCHEMBL14720516

NC(=O)c1ccccc1.c1ccc2ncccc2c1

nearest known ligand 0.61

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.61
CYP3A4 P08684 2/20 0.57
PARP1 P09874 2/20 0.57
POLB P06746 1/20 0.57
MAPT P10636 1/20 0.57
TSHR P16473 1/20 0.57
CYP2C19 P33261 1/20 0.57
RECQL P46063 1/20 0.57
BLM P54132 1/20 0.57
PMP22 Q01453 1/20 0.57
HSD17B10 Q99714 1/20 0.57
TDP1 Q9NUW8 1/20 0.57
L3MBTL1 Q9Y468 1/20 0.57
PABPC1 P11940 1/20 0.51
F7 P08709 1/20 0.47
F3 P13726 1/20 0.47
SARM1 Q6SZW1 1/20 0.47
SIRT2 Q8IXJ6 1/20 0.47
SIRT6 Q8N6T7 1/20 0.47
SIRT1 Q96EB6 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Quinoline SCHEMBL2201840 0.91 ALDH1A1 (0.74) ALDH1A1CYP3A4PARP1POLBMAPT
Quinoline SCHEMBL5272119 0.91 ALDH1A1 (0.74) ALDH1A1CYP3A4PARP1POLBMAPT
8-Aminoquinoline SCHEMBL28879412 0.87 PARP1 (0.50) ALDH1A1CYP3A4PARP1POLBMAPT
Quinoline SCHEMBL29158803 0.87 MEN1 (0.53) ALDH1A1PARP1MAPTCYP2C19TDP1
Quinoline SCHEMBL29158789 0.87 ALDH1A1 (0.53) ALDH1A1CYP3A4PARP1POLBMAPT
Quinoline SCHEMBL1287895 0.87 ALDH1A1 (0.74) ALDH1A1CYP3A4PARP1POLBMAPT
Quinoline SCHEMBL5874527 0.85 ALDH1A1 (0.65) ALDH1A1CYP3A4MAPTTSHRTDP1
Quinoline SCHEMBL8930504 0.85 ALDH1A1 (0.65) ALDH1A1CYP3A4MAPTTSHRTDP1
Quinoxaline SCHEMBL11668022 0.85 MAPT (0.67) ALDH1A1CYP3A4PARP1POLBMAPT
Quinoline SCHEMBL28970061 0.85 ALDH1A1 (0.71) ALDH1A1CYP3A4POLBMAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108752186-A A kind of preparation method of 2- benzyls -5- trifluoromethylbenzoic acids 安徽古尔特科技有限公司 2018-11-06 CN claimed
CN-108485307-A A kind of fluorescent dye, preparation method and applications for opening property with fluorescence 浙江工业大学 2018-09-04 CN disclosed
US-20170349554-A1 COMPOSITIONS AND METHODS FOR TREATING NEURODEGENERATIVE DISEASE COGNITION THERAPEUTICS, INC. 2017-12-07 US disclosed
CN-107260726-A Composition and method for treating nerve degenerative diseases 考格尼申治疗股份有限公司 2017-10-20 CN disclosed
CN-107162972-A The preparation method of the trimethylbenzoyl amine of N phenyl N [8] quinolyl 2,4,6 湖北工业大学 2017-09-15 CN disclosed
CN-106928231-A The kinase inhibitor of the new EGFR wild types of one class and saltant type 合肥中科普瑞昇生物医药科技有限公司 2017-07-07 CN disclosed
US-20140378460-A1 COMPOSITIONS AND METHODS FOR TREATING NEURODEGENERATIVE DISEASE COGNITION THERAPEUTICS, INC. (US) 2014-12-25 US disclosed
CN-104053436-A Compositions and methods for treating neurodegenerative diseases COGNITION THERAPEUTICS INC 2014-09-17 CN disclosed
EP-2747768-A2 COMPOSITIONS AND METHODS FOR TREATING NEURODEGENERATIVE DISEASE Cognition Therapeutics, Inc. (US) 2014-07-02 EP disclosed
CN-103242315-A Salt of quinoline benzamide derivative SHANGHAI YIZHI MEDICAL TECH CO 2013-08-14 CN disclosed
CN-103242315-A Salt of quinoline benzamide derivative SHANGHAI YIZHI MEDICAL TECH CO 2013-08-14 CN disclosed
WO-2013029060-A2 COMPOSITIONS AND METHODS FOR TREATING NEURODEGENERATIVE DISEASE COGNITION THERAPEUTICS, INC. (US) 2013-02-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140378460-A1 COMPOSITIONS AND METHODS FOR TREATING NEURODEGENERATIVE DISEASE TMEM97, SLC18A2, SIGMAR1 ALDH1A1 4387/4885CYP3A4 4754/4885PARP1 4775/4885
US-20170349554-A1 COMPOSITIONS AND METHODS FOR TREATING NEURODEGENERATIVE DISEASE TMEM97, SLC18A2, SIGMAR1 ALDH1A1 4387/4885CYP3A4 4754/4885PARP1 4775/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.