8-Aminoquinoline

8-Aminoquinoline

SCHEMBL28879412

NC(=O)c1ccccc1.Nc1cccc2cccnc12.c1ccc2ncccc2c1

nearest known ligand 0.57

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Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.50
LMNA P02545 2/20 0.47
KDR P35968 1/20 0.47
METAP2 P50579 1/20 0.47
METAP1 P53582 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
ALDH1A1 P00352 4/20 0.46
HDAC1 Q13547 2/20 0.44
HDAC2 Q92769 1/20 0.44
ADORA2A P29274 2/20 0.44
ADORA1 P30542 2/20 0.44
ADORA3 P0DMS8 1/20 0.44
ADORA2B P29275 1/20 0.44
CYP3A4 P08684 2/20 0.43
TDP1 Q9NUW8 2/20 0.43
MAPT P10636 2/20 0.43
POLB P06746 1/20 0.43
TSHR P16473 1/20 0.43
CYP2C19 P33261 1/20 0.43
RECQL P46063 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
8-Aminoquinoline SCHEMBL19748791 0.93 PARP1 (0.57) PARP1LMNAKDRMETAP2METAP1
Quinoline SCHEMBL14720516 0.87 ALDH1A1 (0.61) PARP1KDRALDH1A1HDAC1HDAC2
8-Aminoquinoline SCHEMBL28078884 0.85 ALDH1A1 (0.63) PARP1LMNAMETAP2METAP1ALDH1A1
8-Aminoquinoline SCHEMBL28695606 0.81 L3MBTL1 (0.56) PARP1LMNAKDRALDH1A1HDAC1
8-Aminoquinoline SCHEMBL28223663 0.81 PARP1 (0.53) PARP1LMNAALDH1A1HDAC1TDP1
8-Aminoquinoline SCHEMBL28692373 0.81 KMT2A (0.56) PARP1LMNAMETAP2METAP1HDAC6
Quinoline SCHEMBL5272119 0.79 ALDH1A1 (0.74) PARP1ALDH1A1HDAC1HDAC2CYP3A4
Quinoline SCHEMBL2201840 0.79 ALDH1A1 (0.74) PARP1ALDH1A1HDAC1HDAC2CYP3A4
Quinoline SCHEMBL28083721 0.79 PARP1 (0.81) PARP1LMNAKDRALDH1A1MAPT
8-Aminoquinoline SCHEMBL28214879 0.78 PARP1 (0.59) PARP1LMNAMETAP2METAP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110437148-A A kind of fluorination process of 8- amide groups quinoline HARBIN INST TECHNOLOGY SHENZHEN 2019-11-12 CN disclosed