SCHEMBL14720707

SCHEMBL14720707

CN1CCN(Cc2ccc(C=C3CCN(C(=O)O)CC3)cc2)C1=O

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SRD5A1 P18405 1/20 0.43
LMNA P02545 1/20 0.42
SRD5A2 P31213 6/20 0.41
POLB P06746 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
KMT2A Q03164 1/20 0.39
ALDH1A1 P00352 2/20 0.39
TSHR P16473 1/20 0.39
MCHR1 Q99705 2/20 0.36
GRM2 Q14416 1/20 0.36
OGA O60502 2/20 0.35
ERCC1 P07992 1/20 0.34
ERCC4 Q92889 1/20 0.34
KDM4E B2RXH2 1/20 0.34
CYP3A4 P08684 1/20 0.34
RECQL P46063 1/20 0.34
TDP1 Q9NUW8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14723605 0.85 TP53 (0.46) SRD5A1LMNASRD5A2POLBKMT2A
SCHEMBL14720649 0.79 FKBP1A (0.35) LMNASRD5A2CYP2D6KMT2AALDH1A1
SCHEMBL14720576 0.76 SRD5A1 (0.52) SRD5A1SRD5A2MCHR1OGA
SCHEMBL14720706 0.75 SRD5A1 (0.51) SRD5A1SRD5A2MCHR1OGA
SCHEMBL14722165 0.75 SRD5A1 (0.51) SRD5A1SRD5A2MCHR1OGA
SCHEMBL22683282 0.74 SRD5A1 (0.50) SRD5A1SRD5A2OGATDP1
SCHEMBL14720416 0.74 SRD5A1 (0.48) SRD5A1SRD5A2POLBMCHR1OGA
SCHEMBL17750085 0.73 LSS (0.51) SRD5A1SRD5A2KMT2A
SCHEMBL14722320 0.73 SRD5A1 (0.42) SRD5A1SRD5A2ALDH1A1MCHR1OGA
SCHEMBL14722471 0.73 SRD5A1 (0.42) SRD5A1SRD5A2ALDH1A1MCHR1OGA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013027001-A1 COMPOUNDS AND THEIR USE TO TREAT HISTAMINE H3 RELATED DISORDERS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-02-28 WO disclosed