SCHEMBL14722282

SCHEMBL14722282

CO[C@H]1CCN(Cc2ccc(C=C3CCN(C(C)(C)C)CC3)cc2)C1=O

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PER2 O15055 2/20 0.36
CRY2 Q49AN0 1/20 0.36
SRD5A2 P31213 1/20 0.34
MCHR1 Q99705 1/20 0.34
ACHE P22303 2/20 0.34
SRC P12931 1/20 0.33
ALDH1A1 P00352 1/20 0.33
KCNH2 Q12809 1/20 0.33
AKR1C3 P42330 1/20 0.33
P2RX3 P56373 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14720841 0.87 SRD5A2 (0.35) SRD5A2ALDH1A1KCNH2
SCHEMBL14720825 0.85 TP53 (0.46) SRD5A2ALDH1A1
SCHEMBL14720876 0.84 FKBP1A (0.38) PER2CRY2SRD5A2KCNH2AKR1C3
SCHEMBL14720875 0.84 FKBP1A (0.38) PER2CRY2SRD5A2KCNH2AKR1C3
SCHEMBL14720948 0.75 SRD5A2 (0.39) SRD5A2
SCHEMBL14721350 0.73 HPGD (0.39) SRD5A2MCHR1
SCHEMBL22330321 0.73 FKBP1A (0.49) PER2ALDH1A1
SCHEMBL14722534 0.71 LMNA (0.46) ACHEALDH1A1
SCHEMBL14720708 0.70 SRD5A1 (0.35) SRD5A2MCHR1
SCHEMBL14721266 0.70 SRD5A1 (0.40) SRD5A2MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013027001-A1 COMPOUNDS AND THEIR USE TO TREAT HISTAMINE H3 RELATED DISORDERS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-02-28 WO disclosed