SCHEMBL14720876

SCHEMBL14720876

COC1CCN(Cc2ccc(C=C3CCN(C4CCC4)CC3)cc2)C1=O

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
FKBP1A P62942 1/20 0.38
PER2 O15055 3/20 0.36
SRD5A2 P31213 1/20 0.36
CRY2 Q49AN0 2/20 0.35
AKR1C3 P42330 1/20 0.34
KCNH2 Q12809 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14720875 1.00 FKBP1A (0.38) FKBP1APER2SRD5A2CRY2AKR1C3
SCHEMBL14722282 0.84 PER2 (0.36) PER2SRD5A2CRY2AKR1C3KCNH2
SCHEMBL14720524 0.81 PDE4A (0.35) FKBP1APER2SRD5A2CRY2
SCHEMBL14720525 0.81 PDE4A (0.35) FKBP1APER2SRD5A2CRY2
SCHEMBL14720463 0.80 L3MBTL1 (0.47) SRD5A2KCNH2HRH3
SCHEMBL14721179 0.80 L3MBTL1 (0.50) SRD5A2HRH3
SCHEMBL14720825 0.80 TP53 (0.46) SRD5A2
SCHEMBL14720649 0.79 FKBP1A (0.35) FKBP1ASRD5A2HRH3
SCHEMBL14720643 0.78 OPRM1 (0.41) HRH3
SCHEMBL14722442 0.77 GRM2 (0.47) SRD5A2KCNH2HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013027001-A1 COMPOUNDS AND THEIR USE TO TREAT HISTAMINE H3 RELATED DISORDERS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-02-28 WO claimed
WO-2013027001-A1 COMPOUNDS AND THEIR USE TO TREAT HISTAMINE H3 RELATED DISORDERS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-02-28 WO disclosed