SCHEMBL14722316

SCHEMBL14722316

COc1ccc(C2=CC(O)CCc3c2cc(OC)c(OC)c3OC)cc1NC(=O)O

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
NPSR1 Q6W5P4 1/20 0.35
BTK Q06187 1/20 0.34
TSHR P16473 1/20 0.34
POLB P06746 2/20 0.34
LTB4R Q15722 2/20 0.34
ACLY P53396 1/20 0.34
ALDH1A1 P00352 3/20 0.34
KDM4E B2RXH2 2/20 0.34
LMNA P02545 2/20 0.34
MAPT P10636 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
ABCB1 P08183 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14725525 0.88 BTK (0.37) BTKALDH1A1
SCHEMBL14721210 0.82 KDM4E (0.37) MEN1KMT2ATSHRPOLBLTB4R
SCHEMBL14725387 0.82 EPHX2 (0.38) KMT2A
SCHEMBL14725335 0.82 TUBB4A (0.44)
SCHEMBL14722455 0.82 TUBB4A (0.44)
SCHEMBL14722633 0.81 TUBB4A (0.43)
SCHEMBL14725373 0.81 TUBB4A (0.43)
SCHEMBL14722871 0.80 ACLY (0.34) MEN1KMT2ABTKPOLBLTB4R
SCHEMBL14725383 0.80 TUBB4A (0.43) MEN1KMT2AALDH1A1KDM4ELMNA
SCHEMBL14725310 0.78 MAPK10 (0.38) ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013026942-A1 TUBULIN BINDING AGENTS THE PROVOST, FELLOWS, FOUNDATION SCHOLARS, AND THE OTHER MEMBERS OF BOARD, OF THE COLLEGE OF THE HOLY AND UNDIVIDED TRINITY OF QUEEN ELIZABETH, NEAR DUBLIN (IE) 2013-02-28 WO disclosed