SCHEMBL14725525

SCHEMBL14725525

COc1ccc(C2=CC(O)CCc3c2cc(OC)c(OC)c3OC)cc1NC(=O)OC(C)(C)C

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BTK Q06187 1/20 0.37
ABL1 P00519 7/20 0.34
PTK6 Q13882 5/20 0.34
SRC P12931 3/20 0.33
PIK3CD O00329 1/20 0.33
EGFR P00533 1/20 0.33
KDR P35968 1/20 0.33
PIK3CA P42336 1/20 0.33
PIK3CG P48736 1/20 0.33
BACE1 P56817 1/20 0.33
PRKDC P78527 1/20 0.33
PI4KB Q9UBF8 1/20 0.33
FYN P06241 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.33
AAK1 Q2M2I8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14722316 0.88 MEN1 (0.35) BTKALDH1A1
SCHEMBL14725529 0.84 MMP1 (0.35) ABL1PIK3CDEGFRKDRPIK3CA
SCHEMBL14725391 0.83 SMN1; SMN2 (0.35) BTKABL1PIK3CDEGFRKDR
SCHEMBL14725387 0.81 EPHX2 (0.38)
SCHEMBL14725373 0.79 TUBB4A (0.43)
SCHEMBL14722633 0.79 TUBB4A (0.43)
SCHEMBL14725501 0.78 EPHX2 (0.35) BACE1
SCHEMBL14725519 0.78 TUBB4A (0.37)
SCHEMBL14725502 0.78 TUBB4A (0.37) FYNALDH1A1AAK1
SCHEMBL14722455 0.78 TUBB4A (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013026942-A1 TUBULIN BINDING AGENTS THE PROVOST, FELLOWS, FOUNDATION SCHOLARS, AND THE OTHER MEMBERS OF BOARD, OF THE COLLEGE OF THE HOLY AND UNDIVIDED TRINITY OF QUEEN ELIZABETH, NEAR DUBLIN (IE) 2013-02-28 WO disclosed