SCHEMBL14724688

SCHEMBL14724688

Cc1ccc2nc(C#CCN(C)C)ncc2c1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.37
CYP1A2 P05177 1/20 0.37
ACHE P22303 2/20 0.36
ALDH1A1 P00352 2/20 0.35
NCK1 P16333 1/20 0.35
BACE1 P56817 1/20 0.35
KCNH2 Q12809 3/20 0.34
PKM P14618 1/20 0.33
NOS1 P29475 3/20 0.32
NOS3 P29474 1/20 0.31
NOS2 P35228 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
ITK Q08881 1/20 0.31
PSMB5 P28074 1/20 0.31
NQO2 P16083 1/20 0.31
KDM4E B2RXH2 1/20 0.31
HPGD P15428 1/20 0.31
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5495690 0.84 CYP2A6 (0.36) CYP2A6ALDH1A1BACE1KCNH2
SCHEMBL30718705 0.73 PKM (0.44) CYP2A6CYP1A2ALDH1A1NCK1BACE1
SCHEMBL27141158 0.73 PKM (0.44) CYP2A6CYP1A2ALDH1A1NCK1BACE1
SCHEMBL8404380 0.67 CYP1A2 (0.52) CYP2A6CYP1A2ALDH1A1NCK1BACE1
SCHEMBL14568526 0.67 BRAF (0.43) KCNH2
SCHEMBL19255198 0.66 CYP1A2 (0.43) CYP2A6CYP1A2ALDH1A1NCK1BACE1
SCHEMBL13363088 0.65 CYP1A2 (0.46) CYP2A6CYP1A2ALDH1A1NCK1BACE1
SCHEMBL26337518 0.65 OPRM1 (0.44) CYP1A2ALDH1A1NCK1BACE1MEN1
SCHEMBL18630402 0.64 CYP1A2 (0.48) CYP2A6CYP1A2ALDH1A1NCK1BACE1
SCHEMBL858595 0.64 ALDH1A1 (0.50) CYP2A6CYP1A2ALDH1A1NCK1BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1836174-B1 ARYL NITROGEN-CONTAINING BICYCLIC COMPOUNDS AND THEIR USE AS KINASE INHIBITORS AMGEN INC (US) 2013-02-27 EP disclosed