SCHEMBL147263

SCHEMBL147263

O=C(O)c1ccc2c(c1)[nH]c1ccccc12

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.73
KIF11 P52732 4/20 0.66
HTR7 P34969 1/20 0.60
HTR2B P41595 1/20 0.60
PDPK1 O15530 1/20 0.57
AHR P35869 1/20 0.55
IMPDH2 P12268 2/20 0.55
KDM4E B2RXH2 2/20 0.53
ALDH1A1 P00352 2/20 0.53
GABRP O00591 1/20 0.53
GABRD O14764 1/20 0.53
GABRA1 P14867 1/20 0.53
GABRB1 P18505 1/20 0.53
GABRG2 P18507 1/20 0.53
GABRB3 P28472 1/20 0.53
GABRA5 P31644 1/20 0.53
GABRA3 P34903 1/20 0.53
GABRA2 P47869 1/20 0.53
GABRB2 P47870 1/20 0.53
GABRA4 P48169 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29377098 1.00 PARP1 (0.73) PARP1KIF11HTR7HTR2BPDPK1
SCHEMBL3234597 0.91 PARP1 (0.67) PARP1KIF11HTR7HTR2BPDPK1
Pyridine SCHEMBL27428733 0.91 PARP1 (0.61) PARP1KIF11HTR7HTR2BPDPK1
SCHEMBL23830045 0.90 PARP1 (0.68) PARP1KIF11HTR7HTR2BKDM4E
SCHEMBL29620678 0.90 PARP1 (0.68) PARP1KIF11HTR7HTR2BKDM4E
SCHEMBL70283 0.89 KDM4E (0.60) PARP1KIF11AHRKDM4EALDH1A1
SCHEMBL29823892 0.89 KDM4E (0.60) PARP1KIF11AHRKDM4EALDH1A1
Carbazole SCHEMBL30782024 0.88 ALDH1A1 (0.61) PARP1KIF11AHRKDM4EALDH1A1
Carbazole SCHEMBL28310367 0.88 ALDH1A1 (0.61) PARP1KIF11AHRKDM4EALDH1A1
Hydrochloric Acid SCHEMBL6434116 0.87 KDM4E (0.59) PARP1KIF11HTR7HTR2BAHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 65 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114621752-A Room-temperature phosphorescent waterborne polymer anti-counterfeiting material and preparation method and application thereof 昆明理工大学 2022-06-14 CN claimed
CN-102325752-B Carbazole and carboline kinase inhibitors BRISTOL MYERS SQUIBB CO 2015-02-04 CN claimed
EP-1599202-A1 TETRACYCLIC PYRAZOLE DERIVATIVES AS KINASE INHIBITORS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM Pharmacia Italia S.p.A. (IT) 2005-11-30 EP claimed
WO-2004071507-A1 TETRACYCLIC PYRAZOLE DERIVATIVES AS KINASE INHIBITORS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM PHARMACIA ITALIA S.P.A. (IT) 2004-08-26 WO claimed
WO-1999045926-A1 CONDENSED HETEROCYCLIC COMPOUNDS AS ANTI-INFLAMMATORY AND IMMUNOMODULATORY AGENTS UNIVERSITY COLLEGE CARDIFF CONSULTANTS LIMITED (GB) 1999-09-16 WO claimed
CN-1088209-A Heterogeneous ring compound WELLCOME FOUND (GB) 1994-06-22 CN claimed
JP-61140564-A None JP disclosed
US-20250346585-A1 PHARMACEUTICAL COMPOUNDS FOR THE TREATMENT OF COMPLEMENT MEDIATED DISORDERS ALEXION PHARMACEUTICALS, INC. (US) 2025-11-13 US disclosed
US-20250179046-A1 SEROTONIN 5-HT2B INHIBITORY COMPOUNDS ZOETIS SERVICES LLC 2025-06-05 US disclosed
US-12240827-B2 Serotonin 5-HT2B inhibitory compounds ZOETIS SERVICES LLC (US) 2025-03-04 US disclosed
CN-119364991-A Perovskite solar cell and preparation method thereof 天合光能股份有限公司 2025-01-24 CN disclosed
CN-119364989-A Hole transport layer, perovskite solar cell and preparation method thereof 天合光能股份有限公司 2025-01-24 CN disclosed
EP-3947360-B1 SEROTONIN 5-HT2B INHIBITORY COMPOUNDS ZOETIS SERVICES LLC (US) 2024-08-07 EP disclosed
US-5679694-A LOW TOXICITY AGAINST NORMAL CELL LINES THE WELLCOME FOUNDATION LTD. (GB) 1997-10-21 US disclosed
EP-0741729-A1 ANTITUMOUR TETRACYCLIC COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1996-11-13 EP disclosed
WO-1995021170-A1 ANTITUMOUR TETRACYCLIC COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1995-08-10 WO disclosed
EP-0651750-A1 TETRACYCLIC COMPOUNDS PROCESS AND INTERMEDIATES FOR THEIR PREPARATION AND THEIR USE AS ANTITUMOUR AGENTS THE WELLCOME FOUNDATION LIMITED (GB) 1995-05-10 EP disclosed
CN-1088209-A Heterogeneous ring compound WELLCOME FOUND (GB) 1994-06-22 CN disclosed
JP-S61140564-A CARBAZOLE DERIVATIVE MITSUBISHI CHEM IND LTD 1986-06-27 JP disclosed
US-4009181-A ANTIINFLAMMATORY AGENTS, ANALGESICS, ANTIRHEUMATIC AGENTS HOFFMANN-LA ROCHE INC. (US) 1977-02-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12240827-B2 Serotonin 5-HT2B inhibitory compounds HTR2B, HTR1B, HTR5A PARP1 4048/4885KIF11 3824/4885HTR7 18/4885
US-20250179046-A1 SEROTONIN 5-HT2B INHIBITORY COMPOUNDS HTR2B, HTR1B, HTR5A PARP1 4048/4885KIF11 3824/4885HTR7 18/4885
US-20250346585-A1 PHARMACEUTICAL COMPOUNDS FOR THE TREATMENT OF COMPLEMENT MEDIATED DISORDERS C5, C1S, C9 PARP1 714/4885KIF11 3448/4885HTR7 1298/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.