SCHEMBL14727201

SCHEMBL14727201

C=Cc1ccc(CCCc2ccc(N(c3ccc(CCc4ccc(N(c5ccc(COCc6ccc(C=C)cc6)cc5)c5ccc(-c6ccccc6)cc5)cc4)cc3)c3ccc(-c4ccccc4)cc3)cc2)cc1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.36
AGXT P21549 2/20 0.36
NAAA Q02083 1/20 0.36
HSD11B1 P28845 2/20 0.35
TSHR P16473 1/20 0.35
L3MBTL1 Q9Y468 2/20 0.34
TDP1 Q9NUW8 1/20 0.34
FFAR1 O14842 1/20 0.34
HRH4 Q9H3N8 1/20 0.34
HRH3 Q9Y5N1 1/20 0.34
BCHE P06276 2/20 0.33
POLB P06746 1/20 0.33
GPR84 Q9NQS5 1/20 0.33
HSP90AB1 P08238 1/20 0.33
MAPT P10636 1/20 0.33
LSS P48449 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14727117 0.96 IDO1 (0.39) IDO1AGXTNAAATSHRFFAR1
SCHEMBL14727161 0.92 IDO1 (0.42) IDO1AGXTNAAATSHRPOLB
SCHEMBL14732704 0.91 NAAA (0.43) IDO1AGXTNAAAHSD11B1L3MBTL1
SCHEMBL14727129 0.90 L3MBTL1 (0.40) IDO1AGXTNAAAHSD11B1L3MBTL1
SCHEMBL14727143 0.90 NAAA (0.39) IDO1AGXTNAAATSHRL3MBTL1
SCHEMBL14727131 0.90 NAAA (0.39) IDO1AGXTNAAATSHRL3MBTL1
SCHEMBL13777509 0.89 TSHR (0.41) IDO1AGXTNAAATSHRL3MBTL1
SCHEMBL14727163 0.89 TSHR (0.41) TSHRL3MBTL1TDP1BCHEPOLB
SCHEMBL14727169 0.89 NAAA (0.35) IDO1AGXTNAAATSHRL3MBTL1
SCHEMBL14727152 0.88 HSD11B1 (0.43) HSD11B1TSHRFFAR1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8663883-B2 Charge-transporting film, photoelectric conversion device, electrophotographic photoreceptor, process cartridge, and image forming apparatus FUJI XEROX CO., LTD. (JP) 2014-03-04 US disclosed
US-8663883-B2 Charge-transporting film, photoelectric conversion device, electrophotographic photoreceptor, process cartridge, and image forming apparatus FUJI XEROX CO., LTD. (JP) 2014-03-04 US disclosed
US-20130052570-A1 CHARGE-TRANSPORTING FILM, PHOTOELECTRIC CONVERSION DEVICE, ELECTROPHOTOGRAPHIC PHOTORECEPTOR, PROCESS CARTRIDGE, AND IMAGE FORMING APPARATUS FUJI XEROX CO., LTD. (JP) 2013-02-28 US disclosed
US-20130052570-A1 CHARGE-TRANSPORTING FILM, PHOTOELECTRIC CONVERSION DEVICE, ELECTROPHOTOGRAPHIC PHOTORECEPTOR, PROCESS CARTRIDGE, AND IMAGE FORMING APPARATUS FUJI XEROX CO., LTD. (JP) 2013-02-28 US disclosed