SCHEMBL14733146

SCHEMBL14733146

CSc1cc(C)nc(-c2cccc(CCCc3cccc(-c4cccc(C)n4)n3)n2)n1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.42
CCR8 P51685 1/20 0.42
TGFBR1 P36897 3/20 0.40
KDM4E B2RXH2 1/20 0.37
GRM5 P41594 2/20 0.37
NOS1 P29475 2/20 0.35
NOS2 P35228 2/20 0.35
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
IRAK4 Q9NWZ3 2/20 0.33
KCNH2 Q12809 1/20 0.33
METAP2 P50579 1/20 0.33
NOS3 P29474 1/20 0.33
FFAR1 O14842 4/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14732901 0.89 CCR1 (0.50) CCR1CCR8TGFBR1GRM5NOS1
SCHEMBL14733156 0.83 GRM5 (0.49) CCR1CCR8TGFBR1GRM5KCNH2
SCHEMBL14733132 0.83 CCR1 (0.43) CCR1CCR8TGFBR1GRM5NOS1
SCHEMBL14733135 0.83 LMNA (0.44) CCR1CCR8TGFBR1GRM5NOS1
SCHEMBL14732969 0.81 CCR1 (0.64) CCR1CCR8TGFBR1GRM5NOS1
SCHEMBL14733147 0.81 CCR1 (0.41) CCR1CCR8TGFBR1NOS1NOS2
SCHEMBL14733005 0.79 GRM5 (0.44) CCR1CCR8TGFBR1GRM5FFAR1
SCHEMBL14733134 0.77 CCR1 (0.50) CCR1CCR8TGFBR1KDM4EGRM5
SCHEMBL14732990 0.77 NOS2 (0.49) CCR1CCR8TGFBR1NOS1NOS2
SCHEMBL10369437 0.76 CTSK (0.38) KDM4ENOS1NOS2KCNH2NOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013026866-A2 NOVEL MICROBIOCIDES SYNGENTA PARTICIPATIONS AG (CH) 2013-02-28 WO disclosed