SCHEMBL14733154

SCHEMBL14733154

COc1cc(Br)nc(-c2cccc(C)n2)n1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.48
CCR8 P51685 1/20 0.48
TGFBR1 P36897 5/20 0.41
GAA P10253 2/20 0.41
FFAR1 O14842 1/20 0.37
CYP2A6 P11509 1/20 0.37
METAP2 P50579 1/20 0.37
KDM4E B2RXH2 2/20 0.36
KMT2A Q03164 1/20 0.36
IDH1 O75874 2/20 0.36
MAPK14 Q16539 2/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
CYP1A1 P04798 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP1B1 Q16678 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14721128 0.86 CCR1 (0.60) CCR1CCR8TGFBR1CYP2A6METAP2
SCHEMBL14733155 0.84 CCR1 (0.46) CCR1CCR8TGFBR1GAAFFAR1
SCHEMBL9565637 0.83 RAB9A (0.56) CCR1CCR8TGFBR1GAACYP2A6
SCHEMBL12497117 0.82 CCR1 (0.56) CCR1CCR8TGFBR1CYP2A6METAP2
SCHEMBL10537342 0.80 CCR1 (0.42) CCR1CCR8TGFBR1GAAFFAR1
SCHEMBL10541408 0.78 NPC1 (0.42) CCR1CCR8TGFBR1GAAFFAR1
SCHEMBL10539246 0.78 PDE2A (0.40) CCR1CCR8TGFBR1GAAKDM4E
SCHEMBL14733160 0.77 CCR1 (0.48) CCR1CCR8TGFBR1CYP2A6METAP2
SCHEMBL14733147 0.76 CCR1 (0.41) CCR1CCR8TGFBR1GAAFFAR1
SCHEMBL14732985 0.75 FFAR1 (0.40) CCR1CCR8TGFBR1GAAFFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013026866-A2 NOVEL MICROBIOCIDES SYNGENTA PARTICIPATIONS AG (CH) 2013-02-28 WO disclosed