SCHEMBL14734356

SCHEMBL14734356

Cc1nc2cccc(F)c2nc1C(=O)CBr

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
RAD52 P43351 1/20 0.40
ADORA2A P29274 7/20 0.36
ADORA1 P30542 5/20 0.36
DHODH Q02127 1/20 0.34
PTPN1 P18031 2/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
MAPK1 P28482 1/20 0.33
HTT P42858 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
GSK3B P49841 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14734402 0.82 RAD52 (0.40) RAD52ADORA2AADORA1HTTSMN1; SMN2
SCHEMBL14734375 0.80 MAPT (0.47) PTPN1ALDH1A1LMNAMAPTMAPK1
SCHEMBL15228695 0.74 PTPN1 (0.43) RAD52PTPN1ALDH1A1LMNAMAPT
SCHEMBL14734397 0.74 MAPT (0.44) RAD52ALDH1A1LMNAMAPTMAPK1
SCHEMBL2021969 0.73 CYP1A2 (0.46) RAD52ALDH1A1LMNAMAPTMAPK1
SCHEMBL2131272 0.72 ACHE (0.41) RAD52DHODHALDH1A1LMNAMAPT
SCHEMBL30118358 0.71 PIM1 (0.42) RAD52ALDH1A1LMNAMAPTMAPK1
SCHEMBL15228873 0.69 PTPN1 (0.43) RAD52PTPN1ALDH1A1LMNAMAPT
SCHEMBL14734341 0.68 PIM1 (0.40) RAD52ALDH1A1LMNAMAPTMAPK1
SCHEMBL21857858 0.68 PARP1 (0.40) RAD52ALDH1A1LMNAMAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013027794-A1 NOVEL COMPOUND AND USE THEREOF AS PDE10 INHIBITOR 田辺三菱製薬株式会社 (JP) 2013-02-28 WO disclosed