SCHEMBL14734375

SCHEMBL14734375

Cc1nc2ccccc2nc1C(=O)CBr

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.47
ALDH1A1 P00352 5/20 0.47
SMN1; SMN2 Q16637 4/20 0.47
HTT P42858 3/20 0.45
MAPK1 P28482 2/20 0.45
LMNA P02545 1/20 0.45
KDM4E B2RXH2 3/20 0.43
CYP1A2 P05177 2/20 0.43
PTPN1 P18031 4/20 0.42
GSK3B P49841 3/20 0.42
PDE10A Q9Y233 1/20 0.41
HSD17B10 Q99714 2/20 0.39
TP53 P04637 1/20 0.39
NPC1 O15118 1/20 0.38
EGFR P00533 1/20 0.38
RAB9A P51151 1/20 0.38
HPGD P15428 2/20 0.38
GAA P10253 1/20 0.38
STAT3 P40763 1/20 0.38
NUDT1 P36639 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14734446 0.82 ALDH1A1 (0.47) MAPTALDH1A1SMN1; SMN2HTTMAPK1
SCHEMBL14734356 0.80 RAD52 (0.40) MAPTALDH1A1SMN1; SMN2HTTMAPK1
SCHEMBL4396535 0.79 MAPT (0.52) MAPTALDH1A1SMN1; SMN2HTTMAPK1
SCHEMBL14734437 0.79 MAPT (0.48) MAPTALDH1A1SMN1; SMN2LMNAKDM4E
SCHEMBL2412550 0.78 MAPT (0.43) MAPTALDH1A1SMN1; SMN2HTTMAPK1
SCHEMBL4833903 0.77 MAPT (0.54) MAPTALDH1A1SMN1; SMN2HTTMAPK1
SCHEMBL29670121 0.77 ALDH1A1 (0.72) MAPTALDH1A1SMN1; SMN2HTTMAPK1
SCHEMBL2056931 0.77 ALDH1A1 (0.72) MAPTALDH1A1SMN1; SMN2HTTMAPK1
SCHEMBL6387026 0.76 MAPT (0.52) MAPTALDH1A1SMN1; SMN2HTTMAPK1
SCHEMBL2025252 0.74 LMNA (0.57) MAPTALDH1A1SMN1; SMN2MAPK1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013027794-A1 NOVEL COMPOUND AND USE THEREOF AS PDE10 INHIBITOR 田辺三菱製薬株式会社 (JP) 2013-02-28 WO disclosed