SCHEMBL14743289

SCHEMBL14743289

COC(=O)c1cc(N(C)C(=O)c2cccnc2)c2c(Cl)cc(Cl)cc2c1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.49
GPBAR1 Q8TDU6 5/20 0.46
CYP19A1 P11511 1/20 0.42
CYP11B1 P15538 1/20 0.42
CYP11B2 P19099 1/20 0.42
HSD17B10 Q99714 2/20 0.40
MAPK1 P28482 1/20 0.40
TGM2 P21980 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
RAB9A P51151 5/20 0.39
NPC1 O15118 4/20 0.39
ALOX15 P16050 1/20 0.39
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
TP53 P04637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14743756 0.88 GPBAR1 (0.46) GPBAR1L3MBTL1
SCHEMBL14743805 0.88 GPBAR1 (0.43) ALDH1A1GPBAR1HSD17B10L3MBTL1RAB9A
SCHEMBL14743979 0.87 TSHR (0.42) ALDH1A1GPBAR1L3MBTL1RAB9ANPC1
SCHEMBL14743641 0.85 RAB9A (0.45) GPBAR1HSD17B10L3MBTL1RAB9ANPC1
SCHEMBL14743988 0.83 HTT (0.39) ALDH1A1GPBAR1RAB9ANPC1ALOX15
SCHEMBL14744024 0.82 GPBAR1 (0.42) GPBAR1ALOX15
SCHEMBL14743624 0.80 GPBAR1 (0.38) GPBAR1MAPK1L3MBTL1ALOX15
SCHEMBL14743993 0.79 MAPK1 (0.56) ALDH1A1MAPK1L3MBTL1RAB9ANPC1
SCHEMBL14743411 0.77 TDP1 (0.50) ALDH1A1HSD17B10L3MBTL1NPC1
SCHEMBL14743646 0.77 TSHR (0.43) ALDH1A1L3MBTL1RAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013030358-A1 GLYCINE B ANTAGONISTS MERZ PHARMA GMBH & CO. KGAA (DE) 2013-03-07 WO disclosed