SCHEMBL14746124

SCHEMBL14746124

O=COc1ccc(C(c2ccccc2)(c2ccccc2)[C@H](O)CS)cc1

nearest known ligand 0.32

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 4/20 0.32
CPA3 P15088 1/20 0.32
FOLH1 Q04609 1/20 0.32
KDM4E B2RXH2 6/20 0.32
ALDH1A1 P00352 5/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
GAA P10253 1/20 0.31
PPARG P37231 1/20 0.31
PPARA Q07869 1/20 0.31
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
LMNA P02545 2/20 0.30
POLB P06746 2/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17396368 0.80 CPA3 (0.39) CPA3FOLH1
SCHEMBL14937220 0.80 KIF11 (0.46) KIF11SMN1; SMN2KMT2ALMNA
SCHEMBL14746123 0.80 CPA3 (0.30) CPA3FOLH1
SCHEMBL5703237 0.71 TSHR (0.38) KIF11KDM4EALDH1A1SMN1; SMN2GAA
SCHEMBL13447587 0.71 SMN1; SMN2 (0.49) KDM4EALDH1A1SMN1; SMN2GAAMEN1
SCHEMBL13221992 0.70 ESR1 (0.44) KIF11ALDH1A1MEN1KMT2ALMNA
SCHEMBL9887145 0.68 ESR1 (0.65) KDM4EALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL14169231 0.67 SRD5A2 (0.50) KDM4ESMN1; SMN2KMT2ALMNA
Formic Acid Phenyl Ester SCHEMBL2662 0.67
Formic Acid Phenyl Ester SCHEMBL27326128 0.67 LTA4H (0.45) ALDH1A1GAAPPARGMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3041491-A1 THIOETHER-,ETHER-, AND ALKYLAMINE-LINKED HYDROGEN BOND SURROGATE PERTIDOMIMENTICS New York University (US) 2016-07-13 EP disclosed
WO-2013033645-A1 THIOETHER-,ETHER-, AND ALKYLAMINE-LINKED HYDROGEN BOND SURROGATE PERTIDOMIMENTICS NEW YORK UNIVERSITY (US) 2013-03-07 WO disclosed