SCHEMBL14746159

SCHEMBL14746159

CCc1c(-c2ccc(OC)cc2OC)[nH]c(=O)c(C(=O)O)c1O.CCc1cc(C(=O)O)c(=O)[nH]c1-c1ccc(N2CCCC2)cc1C.CCc1cc(C(=O)O)c(=O)[nH]c1-c1ccc(N2CCCC2)cc1F

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MRGPRX4 Q96LA9 1/20 0.36
KEAP1 Q14145 1/20 0.34
NFE2L2 Q16236 1/20 0.34
MAPT P10636 4/20 0.33
ALDH1A1 P00352 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
RORC P51449 1/20 0.33
DCTPP1 Q9H773 2/20 0.33
THRB P10828 1/20 0.32
USP2 O75604 2/20 0.32
PSMD14 O00487 1/20 0.32
MMP2 P08253 1/20 0.32
PARP1 P09874 1/20 0.32
EDNRB P24530 1/20 0.32
ABCB1 P08183 1/20 0.31
KDM4E B2RXH2 1/20 0.31
POLB P06746 1/20 0.31
GAA P10253 1/20 0.31
HTT P42858 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14746157 0.91 MRGPRX4 (0.35) MRGPRX4KEAP1NFE2L2MAPTALDH1A1
SCHEMBL14745700 0.85 ALDH1A1 (0.34) MAPTALDH1A1L3MBTL1DCTPP1KDM4E
SCHEMBL14746158 0.85 MAPT (0.34) MRGPRX4MAPTALDH1A1L3MBTL1RORC
SCHEMBL14745459 0.81 ABCB1 (0.41) MAPTALDH1A1USP2ABCB1KDM4E
SCHEMBL14745012 0.80 ABCB1 (0.41) KEAP1NFE2L2MAPTALDH1A1L3MBTL1
SCHEMBL14741313 0.80 GRK6 (0.41) MAPTALDH1A1L3MBTL1PARP1KMT2A
SCHEMBL14745359 0.80 PSMD14 (0.38) MRGPRX4MAPTALDH1A1L3MBTL1USP2
SCHEMBL14745409 0.79 GFER (0.39) MRGPRX4MAPTALDH1A1L3MBTL1USP2
SCHEMBL14745493 0.79 ALDH1A1 (0.39) MAPTALDH1A1L3MBTL1USP2KDM4E
SCHEMBL14745618 0.79 ALDH1A1 (0.42) MRGPRX4KEAP1NFE2L2MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2750505-A1 ANTIBACTERIAL COMPOUNDS AND METHODS FOR USE PTC Therapeutics, Inc. (US) 2014-07-09 EP claimed
WO-2013033240-A1 ANTIBACTERIAL COMPOUNDS AND METHODS FOR USE PTC THERAPEUTICS, INC. (US) 2013-03-07 WO claimed