SCHEMBL14747799

SCHEMBL14747799

FC(F)(F)c1nn(-c2ccccc2)c(-c2ccccc2)c1C1CC1

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.47
PTGS1 P23219 3/20 0.47
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
HTR2B P41595 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14747605 0.91 PTGS2 (0.48) PTGS2PTGS1
SCHEMBL6340625 0.86 PTGS2 (0.70) PTGS2PTGS1
SCHEMBL8689472 0.78 PTGS2 (0.47) PTGS2PTGS1
SCHEMBL28617555 0.78 ALDH1A1 (0.41) PTGS2PTGS1
SCHEMBL14747809 0.77 PTGS2 (0.71) PTGS2PTGS1HTR2AHTR2CHTR2B
SCHEMBL14747815 0.76 PTGS2 (0.54) PTGS2PTGS1CYP1A2CYP2C9CYP2C19
SCHEMBL14747800 0.72 PTGS2 (0.50) PTGS2PTGS1CYP1A2CYP2C9CYP2C19
SCHEMBL14747602 0.69 PTGS2 (0.70) PTGS2PTGS1
SCHEMBL29248058 0.68 POLB (0.50) PTGS2PTGS1
SCHEMBL14747603 0.68 PTGS2 (0.55) PTGS2PTGS1CYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE44048-E1 4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyrazol-1-YL]benzenesulfonamide for the treatment of inflammation or an inflammation-associated disorder G.D. SEARLE LLC (US) 2013-03-05 US disclosed