SCHEMBL14747808

SCHEMBL14747808

Fc1cnn(-c2ccccc2)c1-c1ccccc1

nearest known ligand 0.68

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 5/20 0.68
PTGS1 P23219 4/20 0.68
LMNA P02545 4/20 0.50
NPSR1 Q6W5P4 3/20 0.50
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49
S1PR1 P21453 2/20 0.48
ALDH1A1 P00352 3/20 0.47
HTT P42858 2/20 0.46
HIF1A Q16665 2/20 0.46
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
NR3C1 P04150 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14747601 0.88 PTGS2 (0.68) PTGS2PTGS1LMNANPSR1NPC1
SCHEMBL6338986 0.82 PTGS2 (1.00) PTGS2PTGS1
SCHEMBL27333012 0.81 PTGS2 (0.69) PTGS2PTGS1LMNANPC1RAB9A
SCHEMBL7912407 0.78 NPC1 (0.65) PTGS2PTGS1LMNANPC1RAB9A
SCHEMBL31276556 0.78 LMNA (0.58) PTGS2PTGS1LMNANPSR1NPC1
SCHEMBL15779176 0.78 PTGS2 (0.65) PTGS2PTGS1LMNANPSR1NPC1
SCHEMBL31276196 0.77 LMNA (0.56) PTGS2PTGS1LMNANPSR1NPC1
SCHEMBL14747796 0.77 PTGS2 (0.68) PTGS2PTGS1LMNANPSR1NPC1
SCHEMBL14495383 0.77 ALDH1A1 (0.50) PTGS2PTGS1LMNANPSR1NPC1
SCHEMBL22795877 0.77 NPC1 (0.49) PTGS2PTGS1LMNANPSR1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE44048-E1 4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyrazol-1-YL]benzenesulfonamide for the treatment of inflammation or an inflammation-associated disorder G.D. SEARLE LLC (US) 2013-03-05 US disclosed