SCHEMBL14748436

SCHEMBL14748436

Cc1cc(Br)c(C=O)cc1Oc1nc(Cl)ccc1C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKDC P78527 1/20 0.43
LMNA P02545 3/20 0.40
ALDH1A1 P00352 3/20 0.37
MAPT P10636 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
HPGD P15428 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C19 P33261 1/20 0.33
EPAS1 Q99814 1/20 0.33
POLB P06746 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
MPI P34949 1/20 0.32
KMT2A Q03164 1/20 0.32
CRHBP P24387 1/20 0.31
CRHR2 Q13324 1/20 0.31
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14748435 0.83 CRHBP (0.40) PRKDCLMNAALDH1A1MAPTSMN1; SMN2
SCHEMBL19622259 0.82 LMNA (0.41) PRKDCLMNAALDH1A1MAPTSMN1; SMN2
SCHEMBL14748439 0.78 ALDH1A1 (0.38) PRKDCLMNAALDH1A1MAPTSMN1; SMN2
SCHEMBL4253285 0.71 PRKDC (0.75) PRKDCLMNAALDH1A1MAPTSMN1; SMN2
SCHEMBL10102093 0.67 PRKDC (0.53) PRKDCLMNAALDH1A1MAPTSMN1; SMN2
SCHEMBL670086 0.67 LMNA (0.77) PRKDCLMNAALDH1A1MAPTSMN1; SMN2
SCHEMBL20157967 0.67 PRKDC (0.47) PRKDCLMNAALDH1A1MAPTSMN1; SMN2
SCHEMBL10018128 0.66 PRKDC (0.54) PRKDCLMNAALDH1A1MAPTSMN1; SMN2
SCHEMBL19622180 0.65 HAO1 (0.33) PRKDCALDH1A1CYP1A2CYP3A4CYP2C19
SCHEMBL28521484 0.65 PRKDC (0.50) PRKDCLMNAALDH1A1MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2564857-A1 Boron-containing small molecules as anti-inflammatory agents Anacor Pharmaceuticals, Inc. (US) 2013-03-06 EP disclosed