SCHEMBL14757121

SCHEMBL14757121

COc1ccccc1S(=O)(=O)Nc1ccc2c(c1)[nH]c(=O)n2C

nearest known ligand 0.83

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 10/20 0.83
BRD1 O95696 1/20 0.62
BRPF1 P55201 1/20 0.62
PKM P14618 1/20 0.56
CCR4 P51679 2/20 0.56
CREBBP Q92793 1/20 0.55
TP53 P04637 3/20 0.50
BRD2 P25440 1/20 0.50
POLB P06746 1/20 0.49
SLC22A12 Q96S37 1/20 0.49
DDB1 Q16531 1/20 0.47
CRBN Q96SW2 1/20 0.47
TRIM24 O15164 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14722196 0.76 BRPF1 (1.00) BRD4BRD1BRPF1PKMCREBBP
SCHEMBL14721412 0.73 BRD4 (0.67) BRD4BRD1BRPF1PKMCREBBP
SCHEMBL28666833 0.72 BRD4 (0.60) BRD4BRD1BRPF1PKMCREBBP
SCHEMBL7569855 0.71 SLC22A12 (0.58) BRD4BRD1BRPF1PKMCREBBP
SCHEMBL7364604 0.71 CA12 (0.59) BRD4PKMSLC22A12
SCHEMBL29430449 0.71 BRD4 (1.00) BRD4CREBBP
SCHEMBL14721611 0.71 BRD4 (1.00) BRD4CREBBP
SCHEMBL14339623 0.71 LMNA (0.55) BRD4PKMPOLB
SCHEMBL14757111 0.70 BRD4 (0.62) BRD4BRD1BRPF1PKMCREBBP
SCHEMBL5305683 0.70 LMNA (0.66) BRD4PKMTP53SLC22A12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20140243286-A1 BROMODOMAIN LIGANDS CAPABLE OF DIMERIZING IN AN AQUEOUS SOLUTION, AND METHODS OF USING SAME COFERON, INC. (US) 2014-08-28 US disclosed
US-20140243286-A1 BROMODOMAIN LIGANDS CAPABLE OF DIMERIZING IN AN AQUEOUS SOLUTION, AND METHODS OF USING SAME COFERON, INC. (US) 2014-08-28 US disclosed
WO-2013033270-A2 BROMODOMAIN LIGANDS CAPABLE OF DIMERIZING IN AN AQUEOUS SOLUTION, AND METHODS OF USING SAME COFERON, INC. (US) 2013-03-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140243286-A1 BROMODOMAIN LIGANDS CAPABLE OF DIMERIZING IN AN AQUEOUS SOLUTION, AND METHODS OF USING SAME BRDT, BRD4, BRD1 BRD4 2/4885BRD1 3/4885BRPF1 22/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.