SCHEMBL14764291

SCHEMBL14764291

COc1cc(B2OC(C)(C)C(C)(C)O2)cc(C#N)c1C1CC1

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.33
AR P10275 2/20 0.33
CSF1R P07333 1/20 0.32
BCAT1 P54687 1/20 0.31
LPL P06858 1/20 0.31
LIPG Q9Y5X9 1/20 0.31
KDM4E B2RXH2 1/20 0.31
USP2 O75604 1/20 0.31
ALDH1A1 P00352 1/20 0.31
DPP4 P27487 1/20 0.30
ESR2 Q92731 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9947925 0.82 LPL (0.37) ARCSF1RLPLLIPGKDM4E
SCHEMBL16655447 0.80 FPR2 (0.37) CSF1RLPLLIPGKDM4EUSP2
SCHEMBL2656840 0.79 KDM4E (0.40) ARCSF1RLPLLIPGKDM4E
SCHEMBL1668192 0.76 TBK1 (0.39)
SCHEMBL1667913 0.75 ALDH1A1 (0.49) ARCSF1RLPLLIPGKDM4E
SCHEMBL421663 0.75 AR (0.43) ARCSF1RLPLLIPGKDM4E
SCHEMBL2427133 0.73 ESR2 (0.38) LPLLIPGESR2
SCHEMBL21772422 0.73 LPL (0.36) LPLLIPGESR2
SCHEMBL30827381 0.73 LPL (0.36) CSF1RLPLLIPGKDM4EESR2
SCHEMBL20253387 0.73 LPL (0.36) CSF1RLPLLIPGKDM4EESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013034238-A1 BENZONITRILE DERIVATIVES AS KINASE INHIBITORS MERCK PATENT GMBH (DE) 2013-03-14 WO disclosed