SCHEMBL14764299

SCHEMBL14764299

CC(C)(C)OC(=O)ON1CCC(c2cnc(N)nc2)CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DDB1 Q16531 1/20 0.41
CRBN Q96SW2 1/20 0.41
DHFR P00374 1/20 0.35
TRPC6 Q9Y210 3/20 0.34
GPR119 Q8TDV5 4/20 0.34
KDM4E B2RXH2 1/20 0.34
MAPT P10636 1/20 0.34
THRB P10828 1/20 0.34
NAMPT P43490 1/20 0.34
PIK3CA P42336 4/20 0.34
AKT1 P31749 1/20 0.34
MTOR P42345 1/20 0.34
WNT3A P56704 1/20 0.34
HPGDS O60760 2/20 0.33
EGFR P00533 1/20 0.33
LCK P06239 1/20 0.33
JAK3 P52333 1/20 0.33
PIK3R1 P27986 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27964794 0.88 DDB1 (0.39) DDB1CRBNDHFRTRPC6NAMPT
SCHEMBL7303971 0.85 SLC18A3 (0.42) DDB1CRBNGPR119KDM4EMAPT
SCHEMBL15939963 0.81 DDB1 (0.58) DDB1CRBNGPR119KDM4EMAPT
SCHEMBL14764554 0.81 ALOX5AP (0.39) TRPC6GPR119KDM4EMAPTTHRB
SCHEMBL14764202 0.81 TRPC6 (0.51) TRPC6
SCHEMBL14764325 0.79 GPR119 (0.36) DDB1CRBNTRPC6GPR119
SCHEMBL14763960 0.78 GPR119 (0.34) TRPC6GPR119KDM4EMAPTTHRB
SCHEMBL187122 0.76 P2RY14 (0.41) GPR119MAPTNAMPTKMT2A
SCHEMBL14764140 0.76 KDM5A (0.41) DDB1CRBNPIK3CAMTOREGFR
SCHEMBL27900299 0.75 TRPC6 (0.47) DDB1CRBNTRPC6KDM4ENAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013034238-A1 BENZONITRILE DERIVATIVES AS KINASE INHIBITORS MERCK PATENT GMBH (DE) 2013-03-14 WO disclosed