SCHEMBL14764490

SCHEMBL14764490

Cc1nc2c(F)cccc2nc1NN

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.41
MAPT P10636 5/20 0.41
GAA P10253 4/20 0.41
KDM4E B2RXH2 5/20 0.41
RAB9A P51151 3/20 0.41
POLB P06746 1/20 0.41
CRHR1 P34998 2/20 0.36
RAD52 P43351 1/20 0.36
NSD2 O96028 1/20 0.35
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
NPC1 O15118 2/20 0.35
LMNA P02545 2/20 0.35
HPGD P15428 2/20 0.35
MAPK1 P28482 1/20 0.35
PARP1 P09874 1/20 0.34
ILK Q13418 1/20 0.33
PRNP P04156 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14764528 0.93 MAPT (0.41) ALDH1A1MAPTGAAKDM4ERAB9A
SCHEMBL14764362 0.83 MAPT (0.42) ALDH1A1MAPTKDM4ERAB9APOLB
SCHEMBL14764633 0.80 MAPT (0.41) ALDH1A1MAPTKDM4ERAB9APOLB
SCHEMBL14734397 0.80 MAPT (0.44) ALDH1A1MAPTGAAKDM4ERAB9A
SCHEMBL14764689 0.78 NQO2 (0.56) ALDH1A1MAPTGAAKDM4ERAB9A
SCHEMBL12503018 0.76 MAPT (0.58) ALDH1A1MAPTGAAKDM4ERAB9A
SCHEMBL14764430 0.76 MAPT (0.41) ALDH1A1MAPTKDM4ERAB9APOLB
SCHEMBL21857858 0.74 PARP1 (0.40) ALDH1A1MAPTGAAKDM4ERAB9A
SCHEMBL14764585 0.74 TDP1 (0.40) ALDH1A1MAPTGAAKDM4ERAB9A
SCHEMBL14764541 0.73 ALDH1A1 (0.37) ALDH1A1MAPTKDM4ERAB9APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013034758-A1 SUBSTITUTED TRIAZOLOPYRAZINES AND USES THEREOF H. LUNDBECK A/S (DK) 2013-03-14 WO disclosed
WO-2013034755-A1 TRIAZOLOPYRAZINE DERIVATIVES AND THEIR USE FOR TREATING NEUROLOGICAL AND PSYCHIATRIC DISORDERS H. LUNDBECK A/S (DK) 2013-03-14 WO disclosed
WO-2013034755-A1 TRIAZOLOPYRAZINE DERIVATIVES AND THEIR USE FOR TREATING NEUROLOGICAL AND PSYCHIATRIC DISORDERS H. LUNDBECK A/S (DK) 2013-03-14 WO disclosed