SCHEMBL14764844

SCHEMBL14764844

COc1cc(Br)cc2nc(C)c(=O)[nH]c12

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 5/20 0.44
PDE3B Q13370 8/20 0.41
PDE3A Q14432 8/20 0.41
ALDH1A1 P00352 1/20 0.39
PRNP P04156 1/20 0.39
MAPT P10636 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
GRIN2D O15399 3/20 0.38
GRIN3B O60391 3/20 0.38
GRIN1 Q05586 3/20 0.38
GRIN2A Q12879 3/20 0.38
GRIN2B Q13224 3/20 0.38
GRIN2C Q14957 3/20 0.38
GRIN3A Q8TCU5 3/20 0.38
LMNA P02545 1/20 0.35
KMT2A Q03164 1/20 0.35
RNASEH1 O60930 1/20 0.34
CYP19A1 P11511 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16052812 0.84 PDE3B (0.43) NQO2PDE3BPDE3AGRIN2DGRIN3B
SCHEMBL16053154 0.82 PDE3B (0.38) NQO2PDE3BPDE3AGRIN2DGRIN3B
SCHEMBL14765195 0.76 ALDH1A1 (0.45) NQO2PDE3BPDE3AALDH1A1PRNP
SCHEMBL14765103 0.75 NQO2 (0.45) NQO2PDE3BPDE3AALDH1A1MAPT
SCHEMBL31426154 0.73 TYMS (0.34) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL16053360 0.71 XDH (0.39) ALDH1A1MAPTGRIN2DGRIN3BGRIN1
SCHEMBL14765128 0.70 NQO2 (0.42) NQO2PDE3BPDE3AMAPTGRIN2D
SCHEMBL25377211 0.69 DAO (0.35) PDE3BPDE3AGRIN2DGRIN3BGRIN1
SCHEMBL1318287 0.69 RXFP1 (0.37) NQO2PDE3BPDE3AALDH1A1PRNP
SCHEMBL31049738 0.69 DAO (0.35) PDE3BPDE3AGRIN2DGRIN3BGRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014139983-A1 [1,2,4]TRIAZOLO[4,3-A]QUINOXALINES AS DUAL PDE2/PDE10 INHIBITORS H. LUNDBECK A/S (DK) 2014-09-18 WO disclosed
WO-2013034758-A1 SUBSTITUTED TRIAZOLOPYRAZINES AND USES THEREOF H. LUNDBECK A/S (DK) 2013-03-14 WO disclosed
WO-2013034755-A1 TRIAZOLOPYRAZINE DERIVATIVES AND THEIR USE FOR TREATING NEUROLOGICAL AND PSYCHIATRIC DISORDERS H. LUNDBECK A/S (DK) 2013-03-14 WO disclosed