SCHEMBL14764930

SCHEMBL14764930

CCCCCCCCN1CN(c2ccc(N3CCN(c4ccc(O)cc4)CC3)cc2)C=N1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.45
GAA P10253 2/20 0.45
HDAC3 O15379 4/20 0.40
HDAC8 Q9BY41 4/20 0.40
MAPT P10636 3/20 0.39
LMNA P02545 2/20 0.39
ALDH1A1 P00352 2/20 0.38
PKM P14618 1/20 0.38
MIF P14174 1/20 0.38
ME2 P23368 1/20 0.38
ME1 P48163 1/20 0.38
ME3 Q16798 1/20 0.38
S1PR1 P21453 1/20 0.38
GRM2 Q14416 1/20 0.37
PLA2G2A P14555 3/20 0.36
MEN1 O00255 1/20 0.36
MAPK1 P28482 1/20 0.36
KMT2A Q03164 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14764354 0.85 DRD2 (0.51) KDM4EGAAMAPTLMNAALDH1A1
SCHEMBL14765211 0.84 KDM4E (0.44) KDM4EGAAMAPTLMNAALDH1A1
SCHEMBL14764534 0.80 DRD2 (0.53) GAAMAPTLMNAALDH1A1MEN1
SCHEMBL29240322 0.75 KDM4E (0.69) KDM4EGAAMAPTLMNAALDH1A1
SCHEMBL30602861 0.72 MAPT (0.50) KDM4EGAAMAPTLMNAALDH1A1
SCHEMBL10724890 0.70 GAA (0.62) KDM4EGAAMAPTLMNAALDH1A1
Bromide SCHEMBL11215769 0.69 GAA (0.60) KDM4EGAAMAPTLMNAALDH1A1
SCHEMBL30593301 0.69 KDM4E (0.43) KDM4EGAAMAPTLMNAALDH1A1
SCHEMBL14764819 0.69 DRD2 (0.51) GAAMAPTLMNAALDH1A1MAPK1
SCHEMBL15912657 0.68 MAPT (0.58) KDM4EGAAHDAC3HDAC8MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013036866-A1 ITRACONAZOLE ANALOGS AND USE THEREOF THE JOHNS HOPKINS UNIVERSITY (US) 2013-03-14 WO disclosed