SCHEMBL14764819

SCHEMBL14764819

CCN1CN(c2ccc(N3CCN(c4ccc(OC)cc4)CC3)cc2)C=N1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.51
MAPT P10636 6/20 0.48
RAB9A P51151 3/20 0.48
KMT2A Q03164 1/20 0.48
HTR3E A5X5Y0 1/20 0.45
HTR3B O95264 1/20 0.45
ADRB1 P08588 1/20 0.45
HTR3A P46098 1/20 0.45
HTR3D Q70Z44 1/20 0.45
HTR3C Q8WXA8 1/20 0.45
SIGMAR1 Q99720 1/20 0.45
ALDH1A1 P00352 5/20 0.45
GAA P10253 3/20 0.45
HSD17B10 Q99714 1/20 0.45
SMN1; SMN2 Q16637 3/20 0.44
NPC1 O15118 2/20 0.44
L3MBTL1 Q9Y468 2/20 0.43
LMNA P02545 1/20 0.43
TSHR P16473 1/20 0.43
DCTPP1 Q9H773 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14764534 0.87 DRD2 (0.53) DRD2MAPTRAB9AKMT2AHTR3E
SCHEMBL14764354 0.85 DRD2 (0.51) DRD2MAPTRAB9AKMT2AHTR3E
SCHEMBL14765211 0.83 KDM4E (0.44) DRD2MAPTKMT2AALDH1A1GAA
SCHEMBL8353109 0.74 DRD2 (0.75) DRD2MAPTRAB9AKMT2AHTR3E
SCHEMBL28115964 0.72 SIGMAR1 (0.50) MAPTRAB9AKMT2ASIGMAR1ALDH1A1
SCHEMBL8890453 0.72 GAA (0.69) DRD2MAPTRAB9AKMT2AHTR3E
SCHEMBL12265056 0.71 DRD2 (0.65) DRD2MAPTRAB9AKMT2AHTR3E
SCHEMBL5915124 0.68 DRD2 (1.00) DRD2KMT2AHTR3EHTR3BADRB1
SCHEMBL14362730 0.68 HTR3E (0.63) DRD2MAPTRAB9AKMT2AHTR3E
SCHEMBL6153220 0.68 ALDH1A1 (0.66) DRD2MAPTRAB9AKMT2AHTR3E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013036866-A1 ITRACONAZOLE ANALOGS AND USE THEREOF THE JOHNS HOPKINS UNIVERSITY (US) 2013-03-14 WO disclosed