SCHEMBL14765211

SCHEMBL14765211

CCN1CN(c2ccc(N3CCN(c4ccc(O)cc4)CC3)cc2)C=N1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.44
MAPT P10636 5/20 0.44
GAA P10253 5/20 0.44
LMNA P02545 3/20 0.44
ALDH1A1 P00352 3/20 0.44
PKM P14618 1/20 0.44
DRD4 P21917 2/20 0.40
FGFR1 P11362 1/20 0.40
FGFR2 P21802 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
HTT P42858 1/20 0.40
ESR1 P03372 2/20 0.38
ESRRG P62508 2/20 0.38
GFER P55789 2/20 0.37
RAD52 P43351 1/20 0.37
TDP1 Q9NUW8 2/20 0.37
ESRRB O95718 1/20 0.37
ME2 P23368 3/20 0.37
ME1 P48163 3/20 0.37
ME3 Q16798 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14764930 0.84 KDM4E (0.45) KDM4EMAPTGAALMNAALDH1A1
SCHEMBL14764819 0.83 DRD2 (0.51) MAPTGAALMNAALDH1A1SMN1; SMN2
SCHEMBL30602861 0.78 MAPT (0.50) KDM4EMAPTGAALMNAALDH1A1
SCHEMBL30593301 0.75 KDM4E (0.43) KDM4EMAPTGAALMNAALDH1A1
SCHEMBL24452939 0.72 MAPT (0.67) KDM4EMAPTGAALMNAALDH1A1
SCHEMBL7041242 0.71 MAPT (0.68) KDM4EMAPTGAALMNAALDH1A1
SCHEMBL14764534 0.70 DRD2 (0.53) MAPTGAALMNAALDH1A1SMN1; SMN2
SCHEMBL7334978 0.68 CHKA (0.61) KDM4EMAPTGAALMNAALDH1A1
SCHEMBL526167 0.66 ALDH1A1 (0.63) KDM4EMAPTGAALMNAALDH1A1
SCHEMBL10498349 0.66 MAPT (0.62) KDM4EMAPTGAALMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013036866-A1 ITRACONAZOLE ANALOGS AND USE THEREOF THE JOHNS HOPKINS UNIVERSITY (US) 2013-03-14 WO disclosed