SCHEMBL14765002

SCHEMBL14765002

CC1CC(=O)c2ccccc2N1C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR3 P46089 1/20 0.46
NOTUM Q6P988 2/20 0.43
KDM4E B2RXH2 4/20 0.41
ALDH1A1 P00352 4/20 0.41
GAA P10253 2/20 0.41
TTR P02766 1/20 0.40
CES1 P23141 1/20 0.40
HPGD P15428 2/20 0.40
CASP1 P29466 2/20 0.40
HSD17B10 Q99714 2/20 0.40
S100A4 P26447 1/20 0.39
ACHE P22303 1/20 0.39
LMNA P02545 2/20 0.38
GLA P06280 1/20 0.38
TSHR P16473 1/20 0.38
CASP7 P55210 1/20 0.38
KMT2A Q03164 2/20 0.38
EGFR P00533 1/20 0.38
MAPT P10636 1/20 0.38
MAPK1 P28482 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7484240 0.82 MEN1 (0.44) GPR3NOTUMKDM4EALDH1A1GAA
SCHEMBL29866320 0.80 NOTUM (0.42) GPR3NOTUMKDM4EALDH1A1GAA
SCHEMBL10588491 0.80 NOTUM (0.42) NOTUMKDM4EALDH1A1TTRCES1
SCHEMBL27321754 0.78 GPR3 (0.46) GPR3NOTUMKDM4EALDH1A1GAA
SCHEMBL221250 0.76 NOTUM (0.64) NOTUMKDM4EALDH1A1GAACES1
SCHEMBL5835789 0.76 NOTUM (0.64) NOTUMKDM4EALDH1A1GAACES1
SCHEMBL5397337 0.73 LMNA (0.51) NOTUMALDH1A1LMNAKMT2AMEN1
SCHEMBL7733992 0.72 NOTUM (0.55) NOTUMALDH1A1LMNAKMT2AMAPT
SCHEMBL31672940 0.72 NOTUM (0.55) NOTUMALDH1A1LMNAKMT2AMAPT
SCHEMBL6890897 0.72 NOTUM (0.55) NOTUMALDH1A1LMNAKMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111670034-A Pyranopyrazoles and pyrazolopyridines immunomodulators for the treatment of autoimmune diseases 洛克菲勒大学 2020-09-15 CN disclosed
CN-103781783-B The substituted benzothiophene derivative of piperazine as antipsychotic drug 大塚制药株式会社 2016-12-07 CN disclosed
CN-103443092-B As the pyrrole derivative of α 7 cholinocepter conditioning agent LUPIN LTD. (IN) 2015-11-25 CN disclosed
WO-2013035892-A1 PIPERAZINE- SUBSTITUTED BENZOTHIOPHENE DERIVATIVES AS ANTIPSYCHOTIC AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2013-03-14 WO disclosed