SCHEMBL14772007

SCHEMBL14772007

Cc1cc(CI)c(NC(=O)c2nn(C)c3ccccc23)cc1CI

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.50
ROCK1 Q13464 1/20 0.46
HDAC3 O15379 1/20 0.45
HDAC1 Q13547 1/20 0.45
LCK P06239 1/20 0.45
CSK P41240 1/20 0.45
ALDH1A1 P00352 1/20 0.43
CYP3A4 P08684 1/20 0.43
TSHR P16473 1/20 0.43
MAPK1 P28482 1/20 0.43
HSD17B10 Q99714 1/20 0.43
HTR3A P46098 3/20 0.43
HTR3E A5X5Y0 2/20 0.43
HTR3B O95264 2/20 0.43
HTR3D Q70Z44 2/20 0.43
HTR3C Q8WXA8 2/20 0.43
SLC22A2 O15244 1/20 0.42
CHRNB2 P17787 1/20 0.42
CHRNA3 P32297 1/20 0.42
CHRNA4 P43681 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14772006 0.90 KDM4E (0.47) KDM4EROCK1HDAC3HDAC1LCK
SCHEMBL14772008 0.87 KDM4E (0.50) KDM4EROCK1HDAC3HDAC1LCK
SCHEMBL91595 0.80 KDM4E (0.58) KDM4EROCK1HDAC3HDAC1LCK
SCHEMBL14504989 0.79 TSHR (0.48) KDM4EROCK1HDAC3HDAC1LCK
SCHEMBL14772115 0.79 GRM4 (0.39) KDM4ETSHR
SCHEMBL91590 0.78 ALDH1A1 (0.55) KDM4EHDAC3HDAC1LCKCSK
SCHEMBL12327693 0.77 KDM4E (0.46) KDM4EROCK1HDAC3HDAC1LCK
SCHEMBL92358 0.76 KDM4E (0.53) KDM4EROCK1HDAC3HDAC1LCK
SCHEMBL92552 0.76 KDM4E (0.53) KDM4EROCK1HDAC3HDAC1LCK
SCHEMBL91588 0.76 KDM4E (0.53) KDM4EROCK1HDAC3HDAC1LCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130065882-A1 VLA-4 inhibitory drug MACHINAGA NOBUO (JP) 2013-03-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130065882-A1 VLA-4 inhibitory drug VCAM1, ITGB4, ITGA4 KDM4E 996/4885ROCK1 3169/4885HDAC3 432/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.