Clofoctol

Clofoctol

SCHEMBL147809

CC(C)(C)CC(C)(C)c1ccc(O)c(Cc2ccc(Cl)cc2Cl)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 1.00
MEN1 O00255 5/20 1.00
KMT2A Q03164 5/20 1.00
USP2 O75604 3/20 1.00
SMN1; SMN2 Q16637 3/20 1.00
MAPT P10636 3/20 1.00
CASP1 P29466 2/20 1.00
ESR1 P03372 2/20 1.00
TP53 P04637 1/20 1.00
PGR P06401 1/20 1.00
ADORA3 P0DMS8 1/20 1.00
AR P10275 1/20 1.00
DRD1 P21728 1/20 1.00
PTGS1 P23219 1/20 1.00
SLC6A2 P23975 1/20 1.00
PDE4A P27815 1/20 1.00
MAPK1 P28482 1/20 1.00
SLC6A4 P31645 1/20 1.00
OPRM1 P35372 1/20 1.00
DRD3 P35462 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Clofoctol SCHEMBL29397347 1.00 CYP3A4 (1.00) CYP3A4MEN1KMT2AUSP2SMN1; SMN2
SCHEMBL71922 0.85 CYP3A4 (0.73) CYP3A4MEN1KMT2AUSP2SMN1; SMN2
SCHEMBL16656147 0.80 CYP3A4 (0.66) CYP3A4MEN1KMT2AUSP2SMN1; SMN2
SCHEMBL27365508 0.76 CYP3A4 (0.61) CYP3A4MEN1KMT2AUSP2SMN1; SMN2
SCHEMBL9082692 0.76 CYP3A4 (0.60) CYP3A4MEN1KMT2AUSP2SMN1; SMN2
SCHEMBL27365471 0.75 CYP3A4 (0.60) CYP3A4MEN1KMT2AUSP2SMN1; SMN2
SCHEMBL9814995 0.75 KLF10 (0.68) CYP3A4MEN1KMT2AUSP2SMN1; SMN2
SCHEMBL5964677 0.75 CYP3A4 (0.65) CYP3A4MEN1KMT2AUSP2SMN1; SMN2
SCHEMBL8163543 0.74 MAPT (0.59) CYP3A4MEN1KMT2AUSP2SMN1; SMN2
SCHEMBL10802800 0.74 SMN1; SMN2 (0.58) CYP3A4MEN1KMT2AUSP2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1678 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12590963-B2 Anti-cancer treatment of preselected subjects and screening methods to identify susceptible subjects TUDAG TU DRESDEN AKTIENGESELLSCHAFT (DE) 2026-03-31 US claimed
US-20250170082-A1 HPDL INHIBITORS AND USES THEREOF NEW YORK UNIVERSITY (US) 2025-05-29 US claimed
US-12274830-B2 Nitric oxide inhalation therapy for infants with bronchiolitis BEYOND AIR LTD (IL) 2025-04-15 US claimed
WO-2024223624-A1 NEW CLOFOCTOL FORMULATION Institut National de la Santé et de la Recherche Médicale (FR) 2024-10-31 WO claimed
US-20240315965-A1 COMPOSITIONS AND METHODS RELATED TO PHARMACEUTICAL EXCIPIENTS Natural Extraction Systems, LLC (US) 2024-09-26 US claimed
WO-2024189607-A1 METHODS AND BIOAVAILABLE HIGHLY PERMEABLE COMPOUNDS FOR DISEASES TREATMENT DIDENKO KIRILL (MX) 2024-09-19 WO claimed
EP-4164749-B1 COMPOUND AND METHOD FOR THE TREATMENT OF CORONAVIRUSES APTEEUS (FR) 2024-08-07 EP claimed
US-20240238217-A1 USE OF CLOFOCTOL FOR THE TREATMENT OF INFLAMMATION CENTRE HOSPITALIER REGIONAL UNIVERSITAIRE DE LILLE (FR) 2024-07-18 US claimed
US-20240173512-A1 METHODS FOR POTENTIATING ANTIMICROBIAL AGENTS STREETERVILLE CAPITAL, LLC 2024-05-30 US claimed
WO-2024086533-A2 METHODS FOR TREATING OR PREVENTING NEUROENDOCRINE TUMOR FORMATION USING CDC7 INHIBITORS MEMORIAL SLOAN-KETTERING CANCER CENTER (US) 2024-04-25 WO claimed
EP-0786999-A4 COMBINATION METHOD FOR ACNE TREATMENT MERCK & CO INC (US) 1999-01-20 EP claimed
EP-0792371-A4 COMBINATION METHOD FOR ACNE TREATMENT MERCK & CO INC (US) 1998-12-30 EP claimed
US-5811078-A IN A SOLVENT MIXTURE WITH ETHYL OR ISOPROPYL ALCOHOL AND WATER ADOLOR CORPORATION (US) 1998-09-22 US claimed
EP-0852494-A2 PERIPHERALLY ACTIVE ANTI-HYPERALGESIC OPIATES THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1998-07-15 EP claimed
EP-0792371-A1 COMBINATION METHOD FOR ACNE TREATMENT Merck & Co., Inc. (US) 1997-09-03 EP claimed
EP-0786999-A1 COMBINATION METHOD FOR ACNE TREATMENT Merck & Co., Inc. (US) 1997-08-06 EP claimed
WO-1997009973-A2 PERIPHERALLY ACTIVE ANTI-HYPERALGESIC OPIATES THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1997-03-20 WO claimed
US-5543417-A 5 Alpha-reductase inhibitor and at least one of an antibacterial agent, a keratolytic agent or an anti-inflammatory agent MERCK & CO., INC. (US) 1996-08-06 US claimed
WO-1996012487-A1 COMBINATION METHOD FOR ACNE TREATMENT MERCK & CO., INC. (US) 1996-05-02 WO claimed
WO-1996012817-A1 COMBINATION METHOD FOR ACNE TREATMENT MERCK & CO., INC. (US) 1996-05-02 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250170082-A1 HPDL INHIBITORS AND USES THEREOF HPGDS, AIPL1, PON1 CYP3A4 3561/4885MEN1 3237/4885KMT2A 4183/4885
US-12590963-B2 Anti-cancer treatment of preselected subjects and screening methods to identify susceptible subjects TPM4, TPM3, TAGLN2 CYP3A4 171/4885MEN1 2154/4885KMT2A 4500/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.