SCHEMBL14788909

SCHEMBL14788909

CCC1(Cc2ccc([N+](=O)[O-])cc2)C(=O)NC(=O)NC1=O

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.61
MMP8 P22894 5/20 0.50
LMNA P02545 3/20 0.48
MEN1 O00255 1/20 0.46
HTT P42858 1/20 0.46
KMT2A Q03164 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
ALDH1A1 P00352 3/20 0.43
LOXL2 Q9Y4K0 1/20 0.43
MMP2 P08253 4/20 0.42
MMP9 P14780 4/20 0.42
MMP13 P45452 4/20 0.42
METAP1 P53582 1/20 0.42
TSHR P16473 1/20 0.41
HSD17B10 Q99714 1/20 0.41
MAPT P10636 1/20 0.40
IDO1 P14902 1/20 0.40
NR3C1 P04150 1/20 0.39
PGR P06401 1/20 0.39
AR P10275 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL679340 0.71 LOXL2 (0.46) KDM4ELMNAMEN1HTTKMT2A
SCHEMBL27690179 0.71 AKR1B1 (0.51) MEN1KMT2AALDH1A1HSD17B10MAPT
SCHEMBL4507525 0.71 AKR1B1 (0.51) MEN1KMT2AALDH1A1MAPTPGR
SCHEMBL128402 0.69 LOXL2 (0.61) MEN1KMT2ASMN1; SMN2ALDH1A1LOXL2
Barbital SCHEMBL43818 0.69 LMNA (1.00) KDM4EMMP8LMNASMN1; SMN2ALDH1A1
Ammonia Solution, Strong SCHEMBL4739223 0.68 LOXL2 (0.59) MEN1KMT2ASMN1; SMN2ALDH1A1LOXL2
Bromide SCHEMBL2771283 0.68 LOXL2 (0.59) MEN1KMT2ASMN1; SMN2ALDH1A1LOXL2
SCHEMBL14782921 0.68 LMNA (0.47) MMP8LMNAALDH1A1MMP2MMP9
SCHEMBL14782806 0.68 LMNA (0.47) KDM4EMMP8LMNAALDH1A1MMP2
SCHEMBL1204527 0.67 LOXL2 (0.48) KDM4ELMNASMN1; SMN2ALDH1A1LOXL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013038153-A1 18F-LABELLED BARBITURATE COMPOUNDS FOR USE AS POSITRON EMISSION IMAGING AGENTS THE UNIVERSITY COURT OF THE UNIVERSITY OF ABERDEEN (GB) 2013-03-21 WO disclosed