SCHEMBL14818031

SCHEMBL14818031

CN(C)C(=O)CN(C)C(=O)c1ccc(I)cc1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TPMT P51580 1/20 0.41
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HDAC1 Q13547 2/20 0.38
HDAC6 Q9UBN7 2/20 0.38
HIF1A Q16665 1/20 0.37
EPAS1 Q99814 1/20 0.37
DRD2 P14416 1/20 0.37
APP P05067 1/20 0.36
ADORA2A P29274 2/20 0.36
HSD17B1 P14061 1/20 0.36
HSD17B2 P37059 1/20 0.36
GSK3B P49841 1/20 0.36
USP1 O94782 2/20 0.35
CFTR P13569 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15702008 0.84 TPMT (0.42) TPMTCA1CA2ALDH1A1HPGD
SCHEMBL13211865 0.84 MMP13 (0.46) ALDH1A1HPGDSMN1; SMN2HDAC1HDAC6
SCHEMBL12459931 0.82 LMNA (0.44) ALDH1A1HPGDSMN1; SMN2HDAC1HDAC6
SCHEMBL12548024 0.80 KMT2A (0.46) HPGDHDAC1HSD17B1HSD17B2
SCHEMBL643967 0.78 ALDH1A1 (0.59) TPMTCA1CA2ALDH1A1HPGD
SCHEMBL25975198 0.78 HDAC4 (0.49) TPMTCA1CA2HDAC1HDAC6
SCHEMBL27369238 0.76 HDAC4 (0.48) TPMTCA1CA2HDAC1HDAC6
SCHEMBL12547699 0.76 ADORA2A (0.35) ALDH1A1HDAC1HDAC6ADORA2A
SCHEMBL14817910 0.74 PYCR1 (0.49) TPMTCA1CA2HIF1AEPAS1
SCHEMBL12218608 0.73 ESR1 (0.40) CA1CA2HDAC1HDAC6ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1802636-B1 PI3 KINASES INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2013-03-27 EP disclosed