SCHEMBL14844014

SCHEMBL14844014

CC1(C)CNC(=O)N1c1cnc(Br)nc1

nearest known ligand 0.34

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 2/20 0.34
MMP13 P45452 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14843988 0.83 CHRNB2 (0.43) GRM5MMP13
SCHEMBL2560942 0.77 KDM4E (0.37) GRM5
SCHEMBL3785201 0.72 AR (0.55)
SCHEMBL6224475 0.72 MMP13 (0.40) GRM5MMP13
SCHEMBL8306096 0.70 MAPT (0.42)
SCHEMBL14840216 0.70 GRM5 (0.44) GRM5
SCHEMBL2559283 0.70 GRM5 (0.32) GRM5
SCHEMBL16702384 0.69 DDB1 (0.42) GRM5
SCHEMBL2560735 0.67 GRM5 (0.40) GRM5
SCHEMBL16701737 0.67 SIRT6 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2763977-A1 ETHYNYL DERIVATIVES AS MGLUR5 ALLOSTERIC MODULATORS F.HOFFMANN-LA ROCHE AG (CH) 2014-08-13 EP disclosed
WO-2013050454-A1 ETHYNYL DERIVATIVES AS MGLUR5 ALLOSTERIC MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2013-04-11 WO disclosed